SCHEMBL11249009

SCHEMBL11249009

N=C(N)NC(=O)C(Cl)c1c(Cl)cccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
PLAU P00749 1/20 0.35
PLAT P00750 1/20 0.35
GLS O94925 2/20 0.35
AKR1B1 P15121 1/20 0.34
CXCL8 P10145 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
MEN1 O00255 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11249698 0.82 CYP1A2 (0.38) CYP1A2KDM4EALDH1A1LMNAF2
Hydrochloric Acid SCHEMBL11256885 0.77 ALDH1A1 (0.36) CYP1A2KDM4EALDH1A1LMNACXCL8
SCHEMBL7291902 0.76 AKR1B1 (0.42) CYP1A2KDM4EALDH1A1LMNAAKR1B1
SCHEMBL8668403 0.72 MAPT (0.47) KDM4EALDH1A1F2F10PLAU
SCHEMBL29651971 0.71 MAPT (0.53) KDM4EALDH1A1LMNAGPR55MEN1
SCHEMBL11437353 0.70 CYP1A2 (0.42) CYP1A2KDM4EALDH1A1LMNACXCL8
Hydrochloric Acid SCHEMBL7942179 0.70 MAPT (0.46) KDM4EALDH1A1F2F10PLAU
SCHEMBL11247633 0.70 ALDH1A1 (0.48) CYP1A2ALDH1A1LMNAAKR1B1MEN1
SCHEMBL11057728 0.69 CYP1A2 (0.49) CYP1A2KDM4EALDH1A1LMNAMEN1
SCHEMBL11249016 0.69 ADRA2A (0.49) CYP1A2KDM4EALDH1A1LMNAAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4318915-A Substituted guandines and methods of preparation thereof BEIERSDORF AKTIENGESELLSCHAFT (DE) 1982-03-09 US disclosed