SCHEMBL11249698

SCHEMBL11249698

N=C(N)NC(=O)C(Br)c1c(Cl)cccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
KDM4E B2RXH2 4/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
PLAU P00749 1/20 0.34
PLAT P00750 1/20 0.34
CXCL8 P10145 1/20 0.33
ADRA2A P08913 2/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CYP3A4 P08684 1/20 0.32
HTR1A P08908 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
MAOA P21397 1/20 0.32
ADRA1D P25100 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11249009 0.82 CYP1A2 (0.39) CYP1A2KDM4EALDH1A1LMNAF2
SCHEMBL11247962 0.80 GLS (0.40) ALDH1A1LMNAF2F10PLAU
Hydrochloric Acid SCHEMBL11256885 0.76 ALDH1A1 (0.36) CYP1A2KDM4EALDH1A1LMNACXCL8
SCHEMBL11244852 0.73 POLB (0.34) ALDH1A1KMT2AMEN1MAPK1POLB
SCHEMBL11263022 0.73 POLB (0.34) ALDH1A1KMT2AMEN1MAPK1POLB
SCHEMBL11247894 0.71 TSHR (0.42) ALDH1A1CXCL8KMT2AMEN1SLC1A3
SCHEMBL11241971 0.71 ALDH1A1 (0.41) CYP1A2ALDH1A1KMT2AMEN1POLB
SCHEMBL8668403 0.70 MAPT (0.47) KDM4EALDH1A1F2F10PLAU
SCHEMBL11249700 0.70 HTR2B (0.47) CYP1A2KDM4ELMNAADRA2AKMT2A
SCHEMBL5179498 0.70 ALDH1A1 (0.40) CYP1A2ALDH1A1LMNAKMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4318915-A Substituted guandines and methods of preparation thereof BEIERSDORF AKTIENGESELLSCHAFT (DE) 1982-03-09 US disclosed