SCHEMBL7291902

SCHEMBL7291902

NC(=O)C(Cl)c1c(Cl)cccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CXCL8 P10145 1/20 0.39
KMT2A Q03164 3/20 0.39
ADRA2A P08913 2/20 0.39
LMNA P02545 2/20 0.39
CYP2D6 P10635 2/20 0.39
HIF1A Q16665 2/20 0.39
MEN1 O00255 1/20 0.39
CYP3A4 P08684 1/20 0.39
HTR1A P08908 1/20 0.39
CYP2C9 P11712 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
MAOA P21397 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11247633 0.80 ALDH1A1 (0.48) AKR1B1ALDH1A1KMT2ALMNAMEN1
SCHEMBL11249016 0.79 ADRA2A (0.49) AKR1B1ALDH1A1KMT2AADRA2ALMNA
SCHEMBL11040309 0.78 ALDH1A1 (0.41) AKR1B1ALDH1A1CXCL8KMT2AADRA2A
SCHEMBL8830155 0.78 ALDH1A1 (0.41) AKR1B1ALDH1A1CXCL8KMT2AADRA2A
SCHEMBL2838988 0.77 CXCL8 (0.45) ALDH1A1CXCL8KMT2AADRA2ALMNA
SCHEMBL1922886 0.77 HSP90AA1 (0.37) ALDH1A1LMNACYP2D6CYP3A4CYP2C9
SCHEMBL6260569 0.77 CXCL8 (0.53) ALDH1A1CXCL8KMT2AADRA2ALMNA
SCHEMBL11249009 0.76 CYP1A2 (0.39) AKR1B1ALDH1A1CXCL8KMT2AADRA2A
Hydrochloric Acid SCHEMBL4670665 0.74 ADRA2A (0.39) AKR1B1ALDH1A1CXCL8KMT2AADRA2A
SCHEMBL10952785 0.74 GABRA1 (0.43) ALDH1A1LMNAKDM4EPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4567264-A ADRENERGIC BLOCKING AGENTS SYNTEX (U.S.A.) INC. (US) 1986-01-28 US disclosed
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed
EP-0126449-A1 Cardioselective aryloxy- and arylthio-hydroxypropyl piperazinyl acetanilides wich affect calcium entry SYNTEX (U.S.A.) INC. (US) 1984-11-28 EP disclosed