SCHEMBL11260852

SCHEMBL11260852

COC(=O)C(C(C)=O)C(C(=O)c1cccs1)c1ccccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.46
ABCB11 O95342 2/20 0.43
THRB P10828 1/20 0.43
NR1I2 O75469 1/20 0.43
CHRM2 P08172 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2B6 P20813 1/20 0.43
DRD1 P21728 1/20 0.43
HTR2A P28223 1/20 0.43
SLC6A4 P31645 1/20 0.43
CYP2C19 P33261 1/20 0.43
OPRK1 P41145 1/20 0.43
HTR2B P41595 1/20 0.43
KCNH2 Q12809 1/20 0.43
P2RY12 Q9H244 1/20 0.43
TP53 P04637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11266686 0.83 KMT2A (0.50) CYP2C19MAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL11259340 0.81 KMT2A (0.41) OPRM1ABCB11THRBNR1I2CHRM2
SCHEMBL11265313 0.80 HPGD (0.42) L3MBTL1MAPTALDH1A1HPGDTDP1
SCHEMBL11268982 0.76 CYP3A4 (0.40) CYP2C19TP53MAPTALDH1A1HPGD
SCHEMBL6631423 0.71 OPRM1 (0.48) OPRM1ABCB11THRBNR1I2CHRM2
SCHEMBL6631421 0.71 OPRM1 (0.48) OPRM1ABCB11THRBNR1I2CHRM2
SCHEMBL11249228 0.71 ALDH1A1 (0.39) OPRM1ABCB11THRBNR1I2CHRM2
SCHEMBL15163429 0.69 HPGD (0.56) TP53L3MBTL1MAPTALDH1A1HPGD
SCHEMBL3697021 0.68 CASP1 (0.45) OPRM1ABCB11THRBNR1I2CHRM2
Ozone SCHEMBL11388736 0.68 ALDH1A1 (0.36) OPRM1ABCB11THRBNR1I2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4360520-A 1,4-Dihydropyridazine compounds, and their medicinal use BAYER AKTIENGESELLSCHAFT (DE) 1982-11-23 US disclosed