SCHEMBL1126973

SCHEMBL1126973

COCCc1cc(-c2ccccc2C)[nH]c1C(=O)C(=O)Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.40
KDM5A P29375 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
MCL1 Q07820 3/20 0.35
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 2/20 0.34
HSD17B10 Q99714 1/20 0.34
CDC7 O00311 1/20 0.34
MARK3 P27448 1/20 0.34
AXL P30530 1/20 0.34
FRK P42685 1/20 0.34
BLK P51451 1/20 0.34
NEK4 P51957 1/20 0.34
PRKCD Q05655 1/20 0.34
MAP4K2 Q12851 1/20 0.34
CAMK2B Q13554 1/20 0.34
CAMK2G Q13555 1/20 0.34
CAMK2D Q13557 1/20 0.34
CDC42BPA Q5VT25 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1126974 0.67 LMNA (0.43) MCL1ALDH1A1CYP1A2CYP2C19CLK4
SCHEMBL1127376 0.67 LMNA (0.40) MCL1ALDH1A1CYP1A2CYP2C19
SCHEMBL15161899 0.64 ALDH1A1 (0.40) KDM4EALDH1A1
SCHEMBL1156618 0.63 LMNA (0.47) KDM5AKDM4CKDM5BKDM4EALDH1A1
SCHEMBL8816288 0.63 TAAR1 (0.56) KDM4EALDH1A1ALOX5TSHR
SCHEMBL1127778 0.63 LMNA (0.39) MCL1KDM4EALDH1A1CYP1A2CYP2C19
SCHEMBL1127700 0.62 KDM4E (0.40) KDM4EALDH1A1HSD17B10CASP7
SCHEMBL1127138 0.62 PYGL (0.34) ALDH1A1HSD17B10MAP2CYP1A2
SCHEMBL1126976 0.62 JAK3 (0.33)
SCHEMBL9219794 0.62 MAPT (0.36) KDM4EALDH1A1HSD17B10TSHRUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed