SCHEMBL11097656

SCHEMBL11097656

COc1ccc(CN2C3CCC2CC(C(=O)Nc2cc(Cl)c([N+](=O)[O-])cc2OC)C3)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.45
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
TRPV1 Q8NER1 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
CHEK1 O14757 1/20 0.43
LTA4H P09960 1/20 0.42
ALPL P05186 1/20 0.42
ALPI P09923 1/20 0.42
ALPG P10696 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11099758 0.94 CXCR6 (0.46) NPC1RAB9ACHEK1MEN1KMT2A
SCHEMBL11133855 0.93 ALDH1A1 (0.46) NPC1RAB9ACHEK1MEN1KMT2A
SCHEMBL11095527 0.92 CTSD (0.43) NPC1RAB9ACHEK1MEN1KMT2A
SCHEMBL11096572 0.92 DRD2 (0.45) NPC1RAB9AMEN1KMT2A
SCHEMBL11266729 0.85 ACKR3 (0.51) TRPV1MEN1KMT2AALDH1A1MAPT
SCHEMBL11097236 0.85 MAPT (0.45) NPC1RAB9ACHEK1MEN1KMT2A
SCHEMBL11097949 0.85 DRD2 (0.51) CXCR4L3MBTL1LTA4HALPLALPI
SCHEMBL11093919 0.85 UBE2M (0.43) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL11270191 0.84 CXCR4 (0.47) CXCR4L3MBTL1LTA4HALPLALPI
SCHEMBL11089660 0.83 HCRTR1 (0.53) CXCR4MEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP claimed
EP-0031219-B1 ANILINE DERIVATIVES BEECHAM GROUP PLC (GB) 1984-03-07 EP disclosed
US-4350691-A ANTIEMETICS BEECHAM GROUP LIMITED (GB) 1982-09-21 US disclosed
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP disclosed