SCHEMBL11283459

SCHEMBL11283459

COc1cc2c(cc1OCCCN1CCN(c3cccc(Cl)c3)CC1)CCC2

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.60
ABCB1 P08183 3/20 0.58
CHEK1 O14757 2/20 0.57
SIGMAR1 Q99720 1/20 0.56
USP2 O75604 1/20 0.53
LMNA P02545 1/20 0.53
THRB P10828 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11275227 0.89 KCNH2 (0.60) KCNH2ABCB1SIGMAR1LMNA
SCHEMBL11280762 0.88 DRD3 (0.56) SIGMAR1
SCHEMBL11270171 0.87 KCNH2 (0.57) KCNH2ABCB1SIGMAR1LMNA
SCHEMBL11276248 0.87 KCNH2 (0.57) KCNH2ABCB1CHEK1SIGMAR1LMNA
SCHEMBL11300075 0.86 KCNH2 (0.62) KCNH2ABCB1SIGMAR1
SCHEMBL11282244 0.85 DRD2 (0.53) SIGMAR1
SCHEMBL11276199 0.84 KCNH2 (0.58) KCNH2ABCB1SIGMAR1
SCHEMBL11270784 0.84 KCNH2 (0.53) KCNH2ABCB1SIGMAR1LMNA
SCHEMBL11273685 0.83 HTR2A (0.53) LMNA
SCHEMBL11282280 0.83 ADRA1D (0.70) KCNH2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339580-A TRANQUILIZERS, SEDATIVES MITSUBISHI CHEMICAL INDUSTRIES, LIMITED (JP) 1982-07-13 US disclosed
EP-0021368-B1 PIPERAZINYLALKOXYINDANES AND ACID ADDITION SALTS THEREOF MITSUBISHI KASEI CORPORATION (JP) 1982-05-19 EP disclosed
EP-0021368-A1 Piperazinylalkoxyindanes and acid addition salts thereof MITSUBISHI KASEI CORPORATION (JP) 1981-01-07 EP disclosed