SCHEMBL1133097

SCHEMBL1133097

O=Cc1ccoc1B(O)O

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
THRB P10828 1/20 0.35
BLM P54132 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ERN1 O75460 4/20 0.33
TRIM24 O15164 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
CYP2A6 P11509 1/20 0.31
CCR1 P32246 1/20 0.30
CCR5 P51681 1/20 0.30
CCR8 P51685 1/20 0.30
PTPN1 P18031 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22612036 0.71
SCHEMBL7663306 0.71 ALDH1A1 (0.37) ALDH1A1MEN1LMNATHRBBLM
SCHEMBL19138056 0.70 ALDH1A1 (0.44) ALDH1A1MEN1LMNATHRBBLM
SCHEMBL8051718 0.70 ALDH1A1 (0.35) ALDH1A1MEN1LMNATHRBBLM
SCHEMBL5234823 0.70 ALDH1A1 (0.35) ALDH1A1KDM4EMEN1LMNATHRB
SCHEMBL28435187 0.69 ENPP2 (0.30)
SCHEMBL51408 0.69
Water SCHEMBL3454746 0.67 ALDH1A1 (0.41) ALDH1A1MEN1LMNATHRBBLM
SCHEMBL686972 0.67
SCHEMBL1703143 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 128 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013080218-A1 NOVEL INTERMEDIATES AND PROCESS FOR THE PREPARATION OF LAPATINIB AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS FRESENIUS KABI ONCOLOGY LTD. (IN) 2013-06-06 WO claimed
US-20030119178-A1 DNA chip and its preparation SATO KOZO (JP) 2003-06-26 US claimed
US-20010011129-A1 DNA chip and its preparation FUJI PHOTO FILM CO., LTD.; 2001-08-02 US claimed
US-20250388531-A1 SUBSTITUTED TETRACYCLINE COMPOUNDS PARATEK PHARM INNC (US) 2025-12-25 US disclosed
CN-119390732-A Phosphorus-nitrogen synergistic flame-retardant biomass flame retardant and application thereof 常州大学 2025-02-07 CN disclosed
US-20250011292-A1 NOVEL RHODANINE DERIVATIVES AND USES THEREOF GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2025-01-09 US disclosed
EP-4415704-A1 NOVEL RHODANINE DERIVATIVES AND USES THEREOF Georgia State University Research Foundation, Inc. (US) 2024-08-21 EP disclosed
CN-116438153-A Method for producing compound having fluorene skeleton, and compound having fluorene skeleton 帝人株式会社 2023-07-14 CN disclosed
CN-107567443-B Biaryl derivatives as GPR120 agonists 株式会社LG化学 2023-04-28 CN disclosed
WO-2023064368-A1 NOVEL RHODANINE DERIVATIVES AND USES THEREOF GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2023-04-20 WO disclosed
CN-115925679-A Biaryl derivatives as GPR120 agonists 株式会社LG化学 2023-04-07 CN disclosed
EP-1470113-A1 PYRIMIDINONE VIRAL POLYMERASE INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2004-10-27 EP disclosed
US-20040158093-A1 Process for preparing a biaryl compound SUMITOMO CHEMICAL COMPANY, LIMITED 2004-08-12 US disclosed
US-6706703-B2 BIS(5-ARYL-2-PYRIDYL) COMPOUND HAVING EXCELLENT IMMUNOGLOBULIN (IGE) ANTIBODY PRODUCTION INHIBITING ACTIVITY, USEFUL FOR THE PREVENTION OR TREATMENT OF ALLERGIC IMMUNE DISEASES KOWA CO., LTD. (JP) 2004-03-16 US disclosed
US-20040024229-A1 Production method for biarylalanine SUMITOMO CHEMICAL COMPANY, LIMITED 2004-02-05 US disclosed
EP-1346971-A1 Production method for biarylalanine SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2003-09-24 EP disclosed
WO-2003062211-A1 PYRIMIDINONE VIRAL POLYMERASE INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2003-07-31 WO disclosed
US-20030119178-A1 DNA chip and its preparation SATO KOZO (JP) 2003-06-26 US disclosed
US-20030027814-A1 Bis(5-aryl-2-pyridyl) derivatives KOWA CO., LTD. (JP) 2003-02-06 US disclosed
US-20010011129-A1 DNA chip and its preparation FUJI PHOTO FILM CO., LTD.; 2001-08-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040024229-A1 Production method for biarylalanine BCAT2, BCAT1, PAH ALDH1A1 1622/4885KDM4E 987/4885MEN1 443/4885
US-20040158093-A1 Process for preparing a biaryl compound CYP1B1, REL, CYP2F1 ALDH1A1 1099/4885KDM4E 2554/4885MEN1 421/4885
US-20030027814-A1 Bis(5-aryl-2-pyridyl) derivatives AHR, PAH, H1-0 ALDH1A1 868/4885KDM4E 1363/4885MEN1 1195/4885
US-20010011129-A1 DNA chip and its preparation STUB1, DNMT3A, PCNA ALDH1A1 3545/4885KDM4E 769/4885MEN1 3081/4885
US-20250388531-A1 SUBSTITUTED TETRACYCLINE COMPOUNDS TET1, TET3, TRRAP ALDH1A1 3798/4885KDM4E 150/4885MEN1 3139/4885
US-20250011292-A1 NOVEL RHODANINE DERIVATIVES AND USES THEREOF ACE2, RARG, ALAD ALDH1A1 955/4885KDM4E 4281/4885MEN1 2519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.