Water

Water

SCHEMBL3454746

O.O=Cc1ccoc1C=O.O=Cc1ccoc1C=O

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 1/20 0.38
THRB known ✓ P10828 1/20 0.38
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP2A6 P11509 1/20 0.33
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
ERN1 O75460 1/20 0.32
PTPN1 P18031 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
TSHR P16473 1/20 0.31
TRIM24 O15164 1/20 0.31
TRIM33 Q9UPN9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL15210122 1.00 ALDH1A1 (0.41) ALDH1A1MEN1LMNATHRBBLM
SCHEMBL28562323 0.95 ALDH1A1 (0.41) ALDH1A1MEN1LMNATHRBBLM
Dimethylamine SCHEMBL28925370 0.89 ALDH1A1 (0.37) ALDH1A1MEN1LMNATHRBBLM
SCHEMBL3394057 0.81
Furan SCHEMBL29163164 0.80 ALDH1A1 (0.35) ALDH1A1MEN1LMNATHRBBLM
SCHEMBL11306795 0.74 ALDH1A1 (0.33) ALDH1A1
SCHEMBL19138056 0.74 ALDH1A1 (0.44) ALDH1A1MEN1LMNATHRBBLM
Water SCHEMBL27897235 0.73
Water SCHEMBL2308338 0.73 ALDH1A1 (0.34) ALDH1A1LMNATHRBCYP2A6TSHR
SCHEMBL28293969 0.73 MAOB (0.42) ALDH1A1LMNACYP2A6MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233476-B1 Preparation of an ether of 2,5-(hydroxymethyl)furfural (HMF) from a fructose source, an alcohol solvent and an acid catalyst ARCHER DANIELS MIDLAND CO (US) 2013-08-28 EP claimed
EP-2233476-A1 Preparation of an ether of 2,5-(hydroxymethyl)furfural (HMF) from a fructose source, an alcohol solvent and an acid catalyst ARCHER-DANIELS-MIDLAND COMPANY (US) 2010-09-29 EP claimed
US-7579489-B2 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ARCHER-DANIELS-MIDLAND COMPANY (US) 2009-08-25 US claimed
US-20080027236-A1 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ARCHER-DANIELS-MIDLAND COMPANY 2008-01-31 US claimed
EP-1838688-A2 PREPARATION OF 2,5-(HYDROXYMETHYL)FURALDEHYDE (HMF), DERIVATIVES THEREOF AND LEVULINIC ACID FROM FRUCTOSE AS WELL AS PREPARATION OF 2,5-BIS-(HYDROXYMETHYL)FURAN FROM 2,5-(HYDROXYMETHYL)FURALDEHYDE Archer-Daniels-Midland Company (US) 2007-10-03 EP claimed
US-20060142599-A1 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ARCHER -DANIELS- MIDLAND COMPANY 2006-06-29 US claimed
WO-2006063220-A2 PREPARATION OF 2,5-(HYDR0XYMETHYL)FURALDEHYDE (HMF) , DERIVATIVES THEREOF AND LEVULINIC ACID FROM FRUCTOSE AS WELL AS PREPARATION OF 2 , 5-BIS- (HYDROXYMETHYL) FURAN FROM 2 , 5- (HYDROXYMETHYL) FURALDEHYDE ARCHER-DANIELS-MIDLAND COMPANY (US) 2006-06-15 WO claimed
US-9090579-B2 Processes for making sugar and/or sugar alcohol dehydration products ARCHER DANIELS MIDLAND CO. (US) 2015-07-28 US disclosed
US-20150005516-A1 PROCESSES FOR MAKING SUGAR AND/OR SUGAR ALCOHOL DEHYDRATION PRODUCTS ARCHER DANIELS MIDLAND CO (US) 2015-01-01 US disclosed
EP-2233476-B1 Preparation of an ether of 2,5-(hydroxymethyl)furfural (HMF) from a fructose source, an alcohol solvent and an acid catalyst ARCHER DANIELS MIDLAND CO (US) 2013-08-28 EP disclosed
EP-2233476-A1 Preparation of an ether of 2,5-(hydroxymethyl)furfural (HMF) from a fructose source, an alcohol solvent and an acid catalyst ARCHER-DANIELS-MIDLAND COMPANY (US) 2010-09-29 EP disclosed
EP-2233477-A1 Preparation of levulinic acid from fructose using an acid catalyst, a polyethylene glycol and an end-capped polyethylene glycol ARCHER-DANIELS-MIDLAND COMPANY (US) 2010-09-29 EP disclosed
EP-2233478-A1 Preparation of 2,5-bis(hydroxymethyl)furan from 2,5-(hydroxymethyl)furaldehyde to using a nickel-zirconium catalyst ARCHER-DANIELS-MIDLAND COMPANY (US) 2010-09-29 EP disclosed
US-7579489-B2 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ARCHER-DANIELS-MIDLAND COMPANY (US) 2009-08-25 US disclosed
US-20080027236-A1 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ARCHER-DANIELS-MIDLAND COMPANY 2008-01-31 US disclosed
US-7317116-B2 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ARCHER-DANIELS-MIDLAND-COMPANY (US) 2008-01-08 US disclosed
EP-1838688-A2 PREPARATION OF 2,5-(HYDROXYMETHYL)FURALDEHYDE (HMF), DERIVATIVES THEREOF AND LEVULINIC ACID FROM FRUCTOSE AS WELL AS PREPARATION OF 2,5-BIS-(HYDROXYMETHYL)FURAN FROM 2,5-(HYDROXYMETHYL)FURALDEHYDE Archer-Daniels-Midland Company (US) 2007-10-03 EP disclosed
US-20060142599-A1 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ARCHER -DANIELS- MIDLAND COMPANY 2006-06-29 US disclosed
WO-2006063220-A2 PREPARATION OF 2,5-(HYDR0XYMETHYL)FURALDEHYDE (HMF) , DERIVATIVES THEREOF AND LEVULINIC ACID FROM FRUCTOSE AS WELL AS PREPARATION OF 2 , 5-BIS- (HYDROXYMETHYL) FURAN FROM 2 , 5- (HYDROXYMETHYL) FURALDEHYDE ARCHER-DANIELS-MIDLAND COMPANY (US) 2006-06-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060142599-A1 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ALDOA, SORD, DERA MEN1 1591/4885THRB 3651/4885ALDH1A1 65/4885
US-20080027236-A1 Processes for the preparation and purification of hydroxymethylfuraldehyde and derivatives ALDOA, SORD, DERA MEN1 1591/4885THRB 3651/4885ALDH1A1 65/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.