SCHEMBL1134062

SCHEMBL1134062

CC(C)(C)OC(=O)C[N]S(=O)(=O)c1ccc(Oc2ccc(I)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
F2 P00734 2/20 0.39
PRSS1 P07477 2/20 0.39
PRSS2 P07478 2/20 0.39
PRSS3 P35030 2/20 0.39
MMP2 P08253 4/20 0.39
MMP9 P14780 2/20 0.39
POLB P06746 1/20 0.38
MMP13 P45452 5/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 2/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
TBXA2R P21731 4/20 0.36
CA12 O43570 3/20 0.35
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA9 Q16790 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1134049 0.87 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2F2PRSS1PRSS2
SCHEMBL1133836 0.87 MMP13 (0.46) ALDH1A1SMN1; SMN2F2PRSS1PRSS2
SCHEMBL1133821 0.77 SMN1; SMN2 (0.49) ALDH1A1SMN1; SMN2MMP2MMP9POLB
SCHEMBL1133818 0.72 MMP13 (0.44) ALDH1A1SMN1; SMN2MMP2MMP9POLB
SCHEMBL15895195 0.68 PTPN1 (0.50) SMN1; SMN2POLBLMNAMEN1GAA
SCHEMBL25564566 0.65 MMP2 (0.50) ALDH1A1SMN1; SMN2F2PRSS1PRSS2
SCHEMBL1133773 0.65 LMNA (0.59) SMN1; SMN2MMP2MMP9MMP13LMNA
SCHEMBL3669592 0.65 HTT (0.55) ALDH1A1SMN1; SMN2MMP2MMP9POLB
SCHEMBL16447010 0.65 MTNR1A (0.46) SMN1; SMN2LMNA
SCHEMBL2194247 0.64 SMN1; SMN2 (0.49) ALDH1A1SMN1; SMN2MMP2MMP9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2285759-A1 RADIOLABELLED MMP SELECTIVE COMPOUNDS Academisch Medisch Centrum bij de Universiteit van Amsterdam (NL) 2011-02-23 EP disclosed
WO-2009139634-A1 RADIOLABELLED MMP SELECTIVE COMPOUNDS ACADEMISCH MEDISCH CENTRUM BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2009-11-19 WO disclosed
WO-2009139633-A1 RADIOLABELLED MMP SELECTIVE COMPOUNDS ACADEMISCH MEDISCH CENTRUM BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2009-11-19 WO disclosed