SCHEMBL1144892

SCHEMBL1144892

O=C(O)c1cc2c(F)cc(F)cc2[nH]1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EIF4A3 P38919 3/20 0.63
KDM4E B2RXH2 5/20 0.56
HSD17B10 Q99714 4/20 0.56
HPGD P15428 4/20 0.56
LMNA P02545 3/20 0.56
ALDH1A1 P00352 3/20 0.56
CYP2C19 P33261 2/20 0.56
PDPK1 O15530 1/20 0.56
TSHR P16473 1/20 0.56
NFKB1 P19838 1/20 0.56
APEX1 P27695 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
GRIN1 Q05586 2/20 0.51
RHEB Q15382 4/20 0.49
IDO1 P14902 3/20 0.46
TDO2 P48775 3/20 0.46
CNR1 P21554 1/20 0.44
MEN1 O00255 2/20 0.44
MAPK1 P28482 2/20 0.44
KMT2A Q03164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29655546 1.00 EIF4A3 (0.63) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL30536689 0.86 EIF4A3 (0.49) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL24448445 0.85 EIF4A3 (0.47) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL30147573 0.85 EIF4A3 (0.47) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL16234661 0.85 EIF4A3 (0.51) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL30067362 0.85 EIF4A3 (0.47) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL15515831 0.84 GRIN1 (0.70) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL21624049 0.84 KDM4E (0.51) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL20505503 0.84 EIF4A3 (0.54) EIF4A3KDM4EHSD17B10HPGDLMNA
SCHEMBL29974385 0.84 GRIN1 (0.70) EIF4A3KDM4EHSD17B10HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 157 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11718633-B2 Indole compounds, process for the preparation and use thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2023-08-08 US claimed
US-20210238204-A1 INDOLE COMPOUNDS, PROCESS FOR THE PREPARATION AND USE THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2021-08-05 US claimed
US-8242275-B2 Bicyclic pyrazole compounds as antibacterial agents JANSSEN PHARMACEUTICA NV (BE) 2012-08-14 US claimed
US-7842810-B2 2,3-Dihydro-benzo[1,4]dioxine-6-carboxylic acid [2-(6-methoxy-quinolin-4-yl)-4,5,6,7-tetrahydro-2H-indazol-5-yl]-amide JANSSEN PHARMACEUTICA, NV (BE) 2010-11-30 US claimed
US-20100280240-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS ALLISON BRETT D 2010-11-04 US claimed
US-20090023741-A1 ARYL/HETARYLAMIDES AS MODULATORS OF THE EP2 RECEPTOR BAYER SCHERING PHARMA AG (DE) 2009-01-22 US claimed
EP-1863483-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS Janssen Pharmaceutica, N.V. (BE) 2007-12-12 EP claimed
US-20060223810-A1 Bicyclic pyrazole compounds as antibacterial agents JANSSEN PHARMACEUTICA N.V. (BE) 2006-10-05 US claimed
WO-2006105289-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS JANSSEN PHARMACEUTICA N.V. (BE) 2006-10-05 WO claimed
US-20260125366-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS INC (US) 2026-05-07 US disclosed
US-12540141-B2 Spiropyrrolidine derived antiviral agents ENANTA PHARMACEUTICALS, INC. (US) 2026-02-03 US disclosed
EP-4635972-A2 FUNCTIONALIZED PEPTIDES AS ANTIVIRAL AGENTS Enanta Pharmaceuticals, Inc. (US) 2025-10-22 EP disclosed
EP-4612156-A1 ANTI-VIRAL COMPOUNDS Aligos Therapeutics, Inc. (US) 2025-09-10 EP disclosed
EP-4605386-A1 ANTI-VIRAL COMPOUNDS Aligos Therapeutics, Inc. (US) 2025-08-27 EP disclosed
WO-2008152099-A2 ARYL/HETARYLAMIDES AS MODULATORS OF THE EP2 RECEPTOR BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-12-18 WO disclosed
US-20080027122-A1 Indole derivatives TANABE SEIYAKU CO., LTD. 2008-01-31 US disclosed
WO-2008013322-A1 1- (-D-GLYCOPYRANOSYL) - 3 - (4-CYCLOPROPYLPHENYLMETHYL) - 4 - HALOGENO INDOLE DERIVATIVES AND USE THEREOF AS SGLT INHIBITORS. MITSUBISHI TANABE PHARMA CORPORATION (JP) 2008-01-31 WO disclosed
EP-1863483-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS Janssen Pharmaceutica, N.V. (BE) 2007-12-12 EP disclosed
US-20060223810-A1 Bicyclic pyrazole compounds as antibacterial agents JANSSEN PHARMACEUTICA N.V. (BE) 2006-10-05 US disclosed
WO-2006105289-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS JANSSEN PHARMACEUTICA N.V. (BE) 2006-10-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080027122-A1 Indole derivatives SLC5A1, SLC5A2, SLC5A11 EIF4A3 3034/4885KDM4E 1709/4885HSD17B10 750/4885
US-20060223810-A1 Bicyclic pyrazole compounds as antibacterial agents NOD2, BAK1, CASP3 EIF4A3 769/4885KDM4E 4629/4885HSD17B10 3644/4885
US-20100280240-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS NOD2, BAK1, CASP3 EIF4A3 769/4885KDM4E 4629/4885HSD17B10 3644/4885
US-20090023741-A1 ARYL/HETARYLAMIDES AS MODULATORS OF THE EP2 RECEPTOR PTGER2, PTGER1, PTGDR2 EIF4A3 3270/4885KDM4E 3048/4885HSD17B10 297/4885
US-11718633-B2 Indole compounds, process for the preparation and use thereof IDO1, IDO2, INMT EIF4A3 3850/4885KDM4E 1740/4885HSD17B10 1445/4885
US-12540141-B2 Spiropyrrolidine derived antiviral agents ACE2, NR3C2, ACE EIF4A3 352/4885KDM4E 3753/4885HSD17B10 308/4885
US-20210238204-A1 INDOLE COMPOUNDS, PROCESS FOR THE PREPARATION AND USE THEREOF IDO1, IDO2, INMT EIF4A3 3850/4885KDM4E 1740/4885HSD17B10 1445/4885
US-20260125366-A1 METHODS FOR TREATING CANCER AKT2, AKT3, PIK3R5 EIF4A3 528/4885KDM4E 3679/4885HSD17B10 1685/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.