SCHEMBL11469809

SCHEMBL11469809

CN(C)c1ccc(-c2nnc(OCc3ccccc3)nc2-c2ccc(N(C)C)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.47
PIM1 P11309 1/20 0.43
ADK P55263 4/20 0.42
ALDH1A1 P00352 7/20 0.42
NOX1 Q9Y5S8 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAPT P10636 4/20 0.42
HPGD P15428 4/20 0.42
CYP1A2 P05177 4/20 0.41
CYP3A4 P08684 4/20 0.41
HSD17B10 Q99714 4/20 0.41
KDM4E B2RXH2 3/20 0.41
CYP2C19 P33261 3/20 0.41
TP53 P04637 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP2D6 P10635 2/20 0.41
SLC6A3 Q01959 1/20 0.39
MAPK1 P28482 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11709965 0.82 MAPT (0.36) ADKALDH1A1LMNANPSR1MAPT
SCHEMBL11244627 0.81 ADK (0.38) ADKALDH1A1NOX1HTTNPSR1
SCHEMBL11468702 0.81 TP53 (0.49) ALDH1A1LMNAHTTNPSR1MAPT
SCHEMBL11468266 0.79 MAPT (0.36) ADKALDH1A1NOX1MAPTHPGD
SCHEMBL11470140 0.78 TLR7 (0.43) ADKALDH1A1MAPTHPGDCYP3A4
SCHEMBL11485810 0.76 MAPT (0.45) ADKALDH1A1NOX1MAPTHPGD
SCHEMBL11485177 0.74 ADK (0.37) ADKNOX1NPSR1CYP1A2CYP2C19
SCHEMBL11468308 0.73 CYP1A2 (0.37) ADKALDH1A1NOX1LMNAMAPT
SCHEMBL31582507 0.71 HTR7 (0.49) ALDH1A1LMNAHTTNPSR1MAPT
SCHEMBL11273639 0.71 GPR84 (0.49) ALDH1A1LMNANPSR1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4190725-A ANTIINFLAMMATORY ELI LILLY AND COMPANY (US) 1980-02-26 US disclosed
US-4021553-A 5,6-Diaryl-1,2,4-triazines as topically-active anti-inflammatory agents ELI LILLY AND COMPANY (US) 1977-05-03 US disclosed