SCHEMBL1149255

SCHEMBL1149255

O=C(Cl)Cc1cccc(F)c1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.47
SIGMAR1 Q99720 2/20 0.47
SLC1A1 P43005 2/20 0.46
RAB9A P51151 2/20 0.46
IDO1 P14902 2/20 0.46
AGXT P21549 2/20 0.46
CASP3 P42574 1/20 0.46
CASP7 P55210 1/20 0.46
MAPK8 P45983 1/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
KMT2A Q03164 1/20 0.46
SRC P12931 1/20 0.45
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
NR4A2 P43354 2/20 0.45
HCAR2 Q8TDS4 1/20 0.45
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4191880 0.85 CTBP2 (0.44) MEN1KMT2ACES2CES1
SCHEMBL27383159 0.84 TAAR1 (0.47) TAAR1SLC1A1RAB9AIDO1AGXT
SCHEMBL6864466 0.83 TAAR1 (0.50) TAAR1SLC1A1RAB9AIDO1AGXT
SCHEMBL9113 0.82 AKR1B1 (0.58) TAAR1SLC1A1SRCNR4A2HCAR2
SCHEMBL2999227 0.81 VNN1 (0.48) TAAR1SIGMAR1SLC1A1RAB9ACASP3
SCHEMBL1447034 0.81 TAAR1 (0.53) TAAR1SLC1A1CASP3CASP7
SCHEMBL1426756 0.80 MAOB (0.51) TAAR1SLC1A1IDO1AGXTCASP3
SCHEMBL28750039 0.80 MAOB (0.47) TAAR1SLC1A1RAB9AIDO1AGXT
Hydrochloric Acid SCHEMBL2531929 0.80 AKR1B1 (0.56) TAAR1SLC1A1IDO1AGXTSRC
SCHEMBL2029757 0.80 MAPK8 (0.52) TAAR1SLC1A1IDO1AGXTMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 163 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6432953-B1 None US disclosed
US-12435060-B2 Acylamino bridged heterocyclic compound, and composition and application thereof BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2025-10-07 US disclosed
US-12319703-B2 Macrocyclic fused pyrazoles as Mcl-1 inhibitors ASCENTAGE PHARMA (SUZHOU) CO., LTD. (CN) 2025-06-03 US disclosed
CN-119528934-A 2-Pyridothiophene compound, preparation method, application and antitubercular drug thereof 桂林医学院 2025-02-28 CN disclosed
US-12012411-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2024-06-18 US disclosed
WO-2024050825-A1 COMPOUNDS AS MLKL INHIBITORS NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2024-03-14 WO disclosed
EP-3901147-B1 ACYLAMINO BRIDGED HETEROCYCLIC COMPOUND, AND COMPOSITION AND APPLICATION THEREOF BEIJING SCITECH MQ PHARMACEUTICALS LTD (CN) 2023-11-22 EP disclosed
CN-116444521-A Preparation method of chromen-4-one compound and intermediate thereof 同润生物医药(上海)有限公司 2023-07-18 CN disclosed
WO-2023130334-A1 METHOD FOR PREPARING CHROMEN-4-ONE COMPOUND AND INTERMEDIATE THEREOF 同润生物医药(上海)有限公司 2023-07-13 WO disclosed
WO-2023130334-A1 METHOD FOR PREPARING CHROMEN-4-ONE COMPOUND AND INTERMEDIATE THEREOF 同润生物医药(上海)有限公司 2023-07-13 WO disclosed
US-4337250-A NEUROLEPTIC AGENTS PFIZER INC. (US) 1982-06-29 US disclosed
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3992396-A TRANQUILIZERS, HYPNOTICS SANDOZ, INC. (US) 1976-11-16 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12319703-B2 Macrocyclic fused pyrazoles as Mcl-1 inhibitors MCL1, BCL2A1, BCL2L1 TAAR1 3604/4885SIGMAR1 1234/4885SLC1A1 4160/4885
US-12435060-B2 Acylamino bridged heterocyclic compound, and composition and application thereof RIPK1, RIPK3, RIPK4 TAAR1 2621/4885SIGMAR1 3569/4885SLC1A1 1753/4885
US-12012411-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 TAAR1 4764/4885SIGMAR1 3557/4885SLC1A1 4834/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.