SCHEMBL11535382

SCHEMBL11535382

Cc1cc(NC(=O)C2CSc3sccc3C2=O)no1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.44
TDP1 Q9NUW8 3/20 0.44
KMT2A Q03164 7/20 0.44
GAPDH P04406 3/20 0.44
LMNA P02545 1/20 0.43
ALOX15 P16050 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 1/20 0.43
MEN1 O00255 4/20 0.42
MAPT P10636 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
APEX1 P27695 1/20 0.42
PTPN7 P35236 1/20 0.42
RECQL P46063 1/20 0.42
BLM P54132 1/20 0.42
BCL2L1 Q07817 1/20 0.42
MCL1 Q07820 1/20 0.42
PTK2B Q14289 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11534203 0.76 MEN1 (0.45) POLBTDP1KMT2ALMNASMN1; SMN2
SCHEMBL11533101 0.72 KMT2A (0.40) POLBKMT2AGAAMEN1MAPT
SCHEMBL11533430 0.71 HPGD (0.40) ALDH1A1HPGDL3MBTL1HTTNPSR1
SCHEMBL11569730 0.71 ALDH1A1 (0.37) KMT2AMEN1MAPTALDH1A1HPGD
SCHEMBL8833289 0.68 SMN1; SMN2 (0.66) POLBTDP1KMT2ALMNASMN1; SMN2
SCHEMBL11664943 0.66 NPC1 (0.31) ALDH1A1HTT
SCHEMBL2322149 0.63 SMN1; SMN2 (0.59) POLBTDP1KMT2ALMNASMN1; SMN2
SCHEMBL9041665 0.63 SMN1; SMN2 (0.52) KMT2ALMNASMN1; SMN2GAAMEN1
SCHEMBL172042 0.63 MAPT (0.65) KMT2AGAPDHSMN1; SMN2GAAMEN1
SCHEMBL11539690 0.62 KMT2A (0.49) POLBKMT2AGAPDHLMNAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4092325-A 5,6-Dihydro-4-oxo-4H-thieno[2,3-b]thiopyran-5-carboxamides, and process for the preparation thereof WARNER-LAMBERT COMPANY (US) 1978-05-30 US claimed
US-4134900-A 5,6-Dihydro-4-oxo-4H-thieno[2,3-b]thiopyran-5-carboxamides, and process for the preparation thereof WARNER-LAMBERT COMPANY (US) 1979-01-16 US disclosed
US-4134896-A 5,6-Dihydro-4-oxo-4H-thieno[2,3-b]thiopyran-5-carboxamides, and process for the preparation thereof WARNER-LAMBERT COMPANY (US) 1979-01-16 US disclosed
US-4098794-A N-Thiazolyl-5,6-dihydro-4-oxo-4H-thieno[2,3-b]thiopyran-5-carboxamides WARNER-LAMBERT COMPANY (US) 1978-07-04 US disclosed
US-4097441-A 5,6-Dihydro-4-oxo-4H-thieno 2,3-b!thiopyran-5-carboxamides WARNER-LAMBERT COMPANY (US) 1978-06-27 US disclosed
US-4092325-A 5,6-Dihydro-4-oxo-4H-thieno[2,3-b]thiopyran-5-carboxamides, and process for the preparation thereof WARNER-LAMBERT COMPANY (US) 1978-05-30 US disclosed