SCHEMBL1153902

SCHEMBL1153902

FC(F)Oc1cccnc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
CHRNB2 P17787 6/20 0.44
CHRNA4 P43681 6/20 0.44
CHRNB4 P30926 2/20 0.44
CHRNA3 P32297 2/20 0.44
CYP19A1 P11511 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2A6 P11509 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RXRA P19793 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29567546 1.00 LMNA (0.50) LMNATDP1CHRNB2CHRNA4CHRNB4
Formic Acid Methyl Ester SCHEMBL31373300 0.86 KMT2A (0.40) LMNATDP1CHRNB2CHRNA4CHRNB4
Propionic Acid SCHEMBL28238586 0.83 CCNC (0.45) LMNACHRNB2CHRNA4
SCHEMBL29139327 0.83 LMNA (0.47) LMNATDP1CHRNB2CHRNA4CHRNB4
SCHEMBL30297760 0.79 DRD1 (0.33) LMNATDP1ALDH1A1
SCHEMBL28047515 0.79 CYP3A4 (0.54) LMNACYP19A1ALDH1A1CYP1A2CYP3A4
SCHEMBL28760545 0.78 LMNA (0.50) LMNATDP1CHRNB2CHRNA4CHRNB4
SCHEMBL4946642 0.78 CHRNB2 (0.51) LMNATDP1CHRNB2CHRNA4CHRNB4
SCHEMBL29854164 0.78 CHRNB2 (0.51) LMNATDP1CHRNB2CHRNA4CHRNB4
SCHEMBL27732729 0.77 LMNA (0.42) LMNATDP1CHRNB2CHRNA4CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 59 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12545682-B2 Heterocyclic derivatives as P2X7 receptor antagonists BREYE THERAPEUTICS APS (DK) 2026-02-10 US claimed
US-20240034737-A1 Heterocyclic Derivatives as P2X7 Receptor Antagonists BREYE THERAPEUTICS APS (DK) 2024-02-01 US claimed
WO-2022101265-A1 PESTICIDALLY ACTIVE FUSED BICYCLIC HETEROAROMATIC COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2022-05-19 WO claimed
CN-105431420-B Diheteroaryl compounds and uses thereof 豪夫迈·罗氏有限公司 2019-08-13 CN claimed
WO-2016012384-A1 TRIFLUORMETHYLOXAZINE AMIDINES AS BACE1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2016-01-28 WO claimed
EP-4643644-A2 PESTICIDALLY ACTIVE FUSED BICYCLIC HETEROAROMATIC COMPOUNDS Syngenta Crop Protection AG (CH) 2025-11-05 EP disclosed
EP-4069688-B1 PESTICIDALLY ACTIVE FUSED BICYCLIC HETEROAROMATIC AMINO COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2025-10-01 EP disclosed
EP-4051673-B1 PESTICIDALLY ACTIVE FUSED BICYCLIC HETEROAROMATIC COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2025-09-24 EP disclosed
EP-4590397-A1 PCSK9 INHIBITORS AND METHODS OF USE THEREOF Astrazeneca AB (SE) 2025-07-30 EP disclosed
CN-114630825-B Condensed with pesticidal activity bicyclic heteroaromatic compounds 先正达农作物保护股份公司 2025-05-16 CN disclosed
CN-115003666-B Condensed derivatives of pesticidal activity Cyclic heteroaromatic amino compounds 先正达农作物保护股份公司 2025-03-21 CN disclosed
US-20240327397-A1 Pesticidally Active Fused Bicyclic Heteroaromatic Compounds SYNGENTA CROP PROTECTION AG (CH) 2024-10-03 US disclosed
CN-107406462-A Tricyclic DLK inhibitors and uses thereof 豪夫迈·罗氏有限公司 2017-11-28 CN disclosed
CN-106459088-A 2-amino-6-methyl-4,4a,5,6-tetrahydropyrano[3,4-d][1,3]thiazin-8a(8h)-yl-1,3-thiazol-4-yl amides 辉瑞公司 2017-02-22 CN disclosed
CN-105246889-A Fluorinated integrin antagonists SCIFLUOR LIFE SCIENCES LLC 2016-01-13 CN disclosed
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN disclosed
CN-103153963-B Cyclopropane compounds EISAI R&D MAN CO LTD 2014-12-24 CN disclosed
CN-103459384-A Benzoxazepines as inhibitors of PI3K/mTOR and methods of their use and manufacture EXELIXIS INC 2013-12-18 CN disclosed
CN-103153963-A Cyclopropane compounds EISAI R&D MAN CO LTD 2013-06-12 CN disclosed
US-20110039693-A1 Pyrimidylmethyl Sulfonamide Compounds BASF SE (DE) 2011-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240327397-A1 Pesticidally Active Fused Bicyclic Heteroaromatic Compounds DDT, ACHE, GSTO1 LMNA 2238/4885TDP1 1239/4885CHRNB2 576/4885
US-20110039693-A1 Pyrimidylmethyl Sulfonamide Compounds TPMT, NQO2, TST LMNA 3704/4885TDP1 1991/4885CHRNB2 4814/4885
US-20240034737-A1 Heterocyclic Derivatives as P2X7 Receptor Antagonists P2RX7, P2RX3, P2RX1 LMNA 1447/4885TDP1 1868/4885CHRNB2 352/4885
US-12545682-B2 Heterocyclic derivatives as P2X7 receptor antagonists P2RX7, P2RX3, P2RX1 LMNA 1370/4885TDP1 2215/4885CHRNB2 249/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.