SCHEMBL11564440

SCHEMBL11564440

Clc1cc[c]c(-c2c(Cl)cccc2Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.36
TSHR P16473 6/20 0.34
CYP3A4 P08684 3/20 0.34
TDP1 Q9NUW8 2/20 0.34
MAPK1 P28482 1/20 0.34
GABRP O00591 2/20 0.33
GABRD O14764 2/20 0.33
GABRA1 P14867 2/20 0.33
GABRB1 P18505 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA5 P31644 2/20 0.33
GABRA3 P34903 2/20 0.33
GABRA2 P47869 2/20 0.33
GABRB2 P47870 2/20 0.33
GABRA4 P48169 2/20 0.33
GABRE P78334 2/20 0.33
GABRA6 Q16445 2/20 0.33
GABRG1 Q8N1C3 2/20 0.33
GABRG3 Q99928 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2050518 0.80 L3MBTL1 (0.37) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL11566539 0.80 FABP3 (0.33) FABP3FABP4ALDH1A1CYP2A6CYP1A2
SCHEMBL15067608 0.79 TP53 (0.35) TP53TSHRCYP3A4TDP1ALDH1A1
SCHEMBL6682355 0.78 CYP2A6 (0.40) TP53TSHRALDH1A1CYP2A6CYP1A2
SCHEMBL14976333 0.76 RORB (0.38) TP53CYP3A4TDP1MAPK1ALDH1A1
SCHEMBL17999104 0.76 ACHE (0.37) CYP3A4FABP3FABP4ALDH1A1
SCHEMBL3022644 0.75 ALOX5 (0.42) TP53TSHR
SCHEMBL4438343 0.75 TP53 (0.41) TP53TSHRCYP3A4TDP1ALDH1A1
SCHEMBL435005 0.75 AHR (0.45) TP53TSHRCYP3A4ALDH1A1HSD17B10
SCHEMBL436851 0.74 AHR (0.38) TP53TSHRCYP3A4TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2782565-A1 USE OF ARYL AND HETARYL CARBOXAMIDES AS ENDOPARASITICIDES Bayer Intellectual Property GmbH (DE) 2014-10-01 EP disclosed
WO-2013076230-A1 USE OF ARYL AND HETARYL CARBOXAMIDES AS ENDOPARASITICIDES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-05-30 WO disclosed
US-4150158-A Oxadiazindione derivatives useful as insecticides IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1979-04-17 US disclosed