SCHEMBL11626985

SCHEMBL11626985

COc1ccc(CC2(C)CNCCN2C)cc1OC

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.41
SIGMAR1 Q99720 3/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 3/20 0.39
LMNA P02545 2/20 0.39
EBP Q15125 2/20 0.39
MAPK1 P28482 2/20 0.39
HSD17B10 Q99714 2/20 0.39
KDM4E B2RXH2 2/20 0.39
TMEM97 Q5BJF2 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSP90AA1 P07900 1/20 0.38
DHCR7 Q9UBM7 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11630403 0.85 MAPT (0.39) HTTALDH1A1LMNAMAPK1HSD17B10
SCHEMBL11643819 0.76 CYP2D6 (0.41) HTTALDH1A1CYP2D6TSHR
SCHEMBL11645697 0.76 TAAR1 (0.40) HTTALDH1A1MAPK1HSD17B10KDM4E
SCHEMBL11628605 0.74 ALDH1A1 (0.44) CA2SIGMAR1HTTALDH1A1LMNA
SCHEMBL2311298 0.74 CA2 (0.45) CA2SIGMAR1ALDH1A1MAPK1HSD17B10
SCHEMBL6625725 0.71 SIGMAR1 (0.63) SIGMAR1EBPTMEM97
Benderizine SCHEMBL11673167 0.70 ALDH1A1 (0.47) SIGMAR1ALDH1A1EBPTMEM97
Benderizine SCHEMBL1816506 0.70 ALDH1A1 (0.47) SIGMAR1ALDH1A1EBPTMEM97
SCHEMBL29756433 0.70 CYP1A2 (0.57) SIGMAR1ALDH1A1MAPK1KDM4ETSHR
SCHEMBL4324560 0.70 CYP1A2 (0.57) SIGMAR1ALDH1A1MAPK1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031216-A CARDIAC DISEASE, ARRHYTHMIA KNOLL A.G. CHEMISCHE FABRIKEN (DT) 1977-06-21 US claimed
US-4079137-A FOR TREATMENT OF VASCULAR AND CARDIAC DISEASES KNOLL A.G. CHEMISCHE FABRIKEN (DT) 1978-03-14 US disclosed
US-4031216-A CARDIAC DISEASE, ARRHYTHMIA KNOLL A.G. CHEMISCHE FABRIKEN (DT) 1977-06-21 US disclosed
US-3996360-A ANTIARRHYTHMIA KNOLL A.G. CHEMISCHE FABRIKEN (DT) 1976-12-07 US disclosed