SCHEMBL1171673

SCHEMBL1171673

O=C(NC(COCc1ccccc1)C(=O)O)OCc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.64
FOLH1 Q04609 1/20 0.63
PPARG P37231 2/20 0.58
CTSK P43235 4/20 0.57
CTSL P07711 2/20 0.57
CTSS P25774 2/20 0.57
MME P08473 1/20 0.55
TACR1 P25103 2/20 0.54
CTRB1 P17538 2/20 0.54
CTSB P07858 1/20 0.53
IDO1 P14902 1/20 0.53
TDO2 P48775 1/20 0.53
CASP1 P29466 2/20 0.52
ALDH1A1 P00352 1/20 0.52
ALOX15 P16050 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1024175 1.00 PPARA (0.64) PPARAFOLH1PPARGCTSKCTSL
SCHEMBL28595041 1.00 PPARA (0.64) PPARAFOLH1PPARGCTSKCTSL
SCHEMBL5827383 0.94 PPARA (0.62) PPARAFOLH1PPARGCTSKCTSL
SCHEMBL21837541 0.94 PPARA (0.58) PPARAFOLH1PPARGCTSKCTSL
SCHEMBL21837546 0.94 PPARA (0.58) PPARAFOLH1PPARGCTSKCTSL
SCHEMBL7319742 0.91 TACR1 (0.62) CTSKCTSLCTSSTACR1CTSB
SCHEMBL4391662 0.90 PPARA (0.57) PPARAFOLH1PPARGCTSKCTSL
SCHEMBL1170973 0.89 CTSK (0.56) PPARAFOLH1PPARGCTSKCTSL
SCHEMBL31456194 0.89 CTSK (0.60) PPARAFOLH1CTSKCTSLCTSS
SCHEMBL16351361 0.88 KYNU (0.62) PPARACTSKCTSLCTSSTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3672582-B1 COMPOSITIONS AND METHODS FOR TREATING CANCER CEDARS SINAI MEDICAL CENTER (US) 2026-04-15 EP disclosed
US-12421185-B2 Compositions and methods for treating cancer CEDARS-SINAI MEDICAL CENTER (US) 2025-09-23 US disclosed
US-11529338-B2 Compositions and methods for treating cancer CEDARS-SINAI MEDICAL CENTER (US) 2022-12-20 US disclosed
CN-115053184-A Composition for forming EUV resist underlayer film 日产化学株式会社 2022-09-13 CN disclosed
CN-107709301-B Pyrazole derivative or pharmacologically acceptable salt thereof 橘生药品工业株式会社 2021-06-22 CN disclosed
US-20210163403-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER CEDARS-SINAI MEDICAL CENTER (US) 2021-06-03 US disclosed
US-10927070-B2 Compositions and methods for treating cancer CEDARS-SINAI MEDICAL CENTER (US) 2021-02-23 US disclosed
US-20200188373-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER CEDARS-SINAI MEDICAL CENTER (US) 2020-06-18 US disclosed
EP-3319970-B1 PYRIDO-OXAZINONE DERIVATIVES AS TNAP INHIBITORS DAIICHI SANKYO CO LTD (JP) 2019-08-28 EP disclosed
US-20190194124-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER CEDARS-SINAI MEDICAL CENTER (US) 2019-06-27 US disclosed
EP-1147095-B1 2, 3, 4, 5-TETRAHYDRO-1H-[1, 4] BENZODIAZEPINE-3-HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS WYETH CORP (US) 2004-08-11 EP disclosed
US-6544984-B1 Treating disease conditions mediated by matrix metalloproteinases and TACE, such as tumor growth, osteoarthritis, rheumatoid arthritis and degenerative cartilage loss. AMERICAN CYANAMID COMPANY 2003-04-08 US disclosed
EP-1147095-A1 2, 3, 4, 5-TETRAHYDRO-1H-[1, 4] BENZODIAZEPINE-3-HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS American Cyanamid Company (US) 2001-10-24 EP disclosed
CN-1293663-A 2,3,4,5-tetrahydro-1H-[1,4] benzodiazepine-3-hydroxamix acids as matrix metal-protease AMERICAN CYANAMID CO (US) 2001-05-02 CN disclosed
EP-1051407-A1 2,3,4,5-TETRAHYDRO-1H-[1,4]-BENZODIAZEPINE-3-HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS American Cyanamid Company (US) 2000-11-15 EP disclosed
WO-2000044730-A1 2,3,4,5-TETRAHYDRO-1H-[1,4]BENZODIAZEPINE-3-HYDROXAMIC ACID AS MATRIX METALLOPROTEINASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-08-03 WO disclosed
US-6071903-A ENZYME INHIBITORS OF MATRIX METALLOPROTEINASES (MMPS); ANTITUMOR,-CARCINOGENIC AND -ARTHRITIC AGENTS; OSTEOARTHRITIS; RHEUMATOID DISEASES; DEGENERATIVE CARTILAGE LOSS; LONG-ACTING, ORALLY BIOAVAILABLE NONPEPTIDE INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-06-06 US disclosed
WO-1999037625-A1 2,3,4,5-TETRAHYDRO-1H-[1,4]-BENZODIAZEPINE-3-HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1999-07-29 WO disclosed
US-4564471-A N-/BENZYLOXYCARBONYL/ASPARTYLPHENYLALANINE AJINOMOTO CO., INC. (JP) 1986-01-14 US disclosed
EP-0027319-A2 Method for reductive elimination of protecting groups and preparative process using such method AJINOMOTO CO., INC. (JP) 1981-04-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12421185-B2 Compositions and methods for treating cancer TSG101, RNASE1, TP53 PPARA 2140/4885FOLH1 25/4885PPARG 1746/4885
US-20210163403-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER TSG101, RNASE1, TP53 PPARA 2140/4885FOLH1 25/4885PPARG 1746/4885
US-11529338-B2 Compositions and methods for treating cancer CHRNB2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, NNMT PPARA 3070/4885FOLH1 416/4885PPARG 2340/4885
US-20200188373-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER CHRNB2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, NNMT PPARA 3070/4885FOLH1 416/4885PPARG 2340/4885
US-20190194124-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER TSG101, TP53, RNASE1 PPARA 2218/4885FOLH1 55/4885PPARG 1924/4885
US-10927070-B2 Compositions and methods for treating cancer TSG101, RNASE1, TP53 PPARA 2140/4885FOLH1 25/4885PPARG 1746/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.