SCHEMBL11757957

SCHEMBL11757957

O=C(Nc1ccc(S(=O)(=O)[O-])c2cccc(S(=O)(=O)[O-])c12)c1ccc([N+](=O)[O-])cc1.[Na+].[Na+]

nearest known ligand 0.57

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DUSP3 P51452 1/20 0.57
PTPN5 P54829 1/20 0.57
CASP6 P55212 1/20 0.57
PTPN11 Q06124 1/20 0.57
CD40 P25942 3/20 0.54
CD40LG P29965 3/20 0.54
PARP1 P09874 1/20 0.52
F11 P03951 1/20 0.51
MAPT P10636 6/20 0.49
KMT2A Q03164 4/20 0.49
TDP1 Q9NUW8 4/20 0.49
ALDH1A1 P00352 3/20 0.49
LMNA P02545 3/20 0.49
POLB P06746 3/20 0.49
PKM P14618 3/20 0.49
TSHR P16473 3/20 0.49
NFKB1 P19838 3/20 0.49
APEX1 P27695 3/20 0.49
RECQL P46063 3/20 0.49
P2RX1 P51575 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11762070 0.89 KMT2A (0.57) DUSP3PTPN5PTPN11MAPTKMT2A
SCHEMBL11757962 0.86 CD40 (0.66) DUSP3PTPN5CASP6PTPN11CD40
SCHEMBL11438902 0.86 KMT2A (0.45) DUSP3PTPN5CASP6PTPN11CD40
SCHEMBL11758753 0.85 SIRT2 (0.55) F11MAPTKMT2ATDP1ALDH1A1
SCHEMBL11432355 0.81 CD40 (0.63) DUSP3PTPN5CASP6PTPN11CD40
SCHEMBL11425283 0.81 CD40 (0.64) DUSP3PTPN5CASP6PTPN11CD40
SCHEMBL11212272 0.81 NPC1 (0.57) DUSP3PTPN5PTPN11MAPTKMT2A
SCHEMBL11421827 0.79 CD40 (0.63) DUSP3PTPN5CASP6PTPN11CD40
SCHEMBL11431112 0.79 CD40 (0.61) DUSP3PTPN5CASP6PTPN11CD40
SCHEMBL11758251 0.78 SIRT2 (0.64) F11MAPTKMT2ATDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4027038-A NAPHTHALENEDISULFONIC ACID UREIDES AMERICAN CYANAMID COMPANY (US) 1977-05-31 US disclosed