SCHEMBL11824198

SCHEMBL11824198

Cc1nccn1-c1nc(Cl)cc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.40
CYP2E1 P05181 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
BDKRB2 P30411 1/20 0.38
MAPT P10636 1/20 0.37
ATM Q13315 1/20 0.37
GRM5 P41594 1/20 0.36
ALDH1A1 P00352 2/20 0.35
KDR P35968 1/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
MAPK9 P45984 1/20 0.34
MAPK10 P53779 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11822572 0.83 KDR (0.44) KDRMAPK9MAPK10
SCHEMBL11818894 0.82 TSHR (0.40) MAPTLMNAHRH4
SCHEMBL11816596 0.77 CYP1A2 (0.43) CYP2A6MAPTALDH1A1LMNAHRH4
SCHEMBL11817340 0.73 MAOA (0.41) CYP2A6CYP2E1CYP3A4MAOAMAOB
SCHEMBL9405397 0.70 NPC1 (0.49) CYP2A6CYP2E1CYP3A4MAOAMAOB
SCHEMBL11814264 0.70 CYP3A4 (0.52) CYP3A4MAPTALDH1A1LMNA
SCHEMBL11820380 0.70 MKNK1 (0.35) ATM
SCHEMBL8498623 0.68 CYP3A4 (0.50) CYP2A6CYP2E1CYP3A4GRM5ALDH1A1
SCHEMBL2170888 0.68 CYP2A6 (0.47) CYP2A6MAPTALDH1A1LMNA
SCHEMBL11816652 0.68 GABRG2 (0.36) MAPTATMALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3961062-A Pharmaceutical composition containing 1-(imidazole-1-yl)-isoquinolines and method of treating hyperlipemia HOECHST AKTIENGESELLSCHAFT (DT) 1976-06-01 US disclosed