SCHEMBL119616

SCHEMBL119616

O=C(O)CN(c1cccc(C(F)(F)F)c1)S(=O)(=O)c1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.72
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
HPGD P15428 1/20 0.62
HTT P42858 1/20 0.62
RORC P51449 9/20 0.59
KEAP1 Q14145 2/20 0.58
NFE2L2 Q16236 2/20 0.58
ALDH1A1 P00352 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7828272 0.90 L3MBTL1 (0.62) L3MBTL1MEN1KMT2AHPGDHTT
SCHEMBL24279586 0.90 MEN1 (0.60) L3MBTL1MEN1KMT2AHPGDHTT
SCHEMBL1631811 0.87 KEAP1 (0.66) L3MBTL1RORCKEAP1NFE2L2
SCHEMBL121206 0.86 RORC (0.70) HPGDHTTRORCALDH1A1
SCHEMBL120825 0.85 HPGD (0.61) L3MBTL1MEN1KMT2AHPGDHTT
SCHEMBL27849029 0.85 HPGD (0.72) L3MBTL1MEN1KMT2AHPGDHTT
SCHEMBL119929 0.84 RORC (0.79) MEN1KMT2AHPGDHTTRORC
SCHEMBL120536 0.83 HTT (0.75) L3MBTL1MEN1KMT2AHPGDHTT
SCHEMBL30458040 0.82 RORC (0.68) MEN1KMT2AHTTRORCALDH1A1
SCHEMBL702692 0.81 KEAP1 (0.68) L3MBTL1KEAP1NFE2L2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102427810-A Sulfamoylbenzoic acid derivatives as TRPM8 antagonists RAQUALIA PHARMA INC 2012-04-25 CN disclosed
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
EP-2424517-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RaQualia Pharma Inc (JP) 2012-03-07 EP disclosed
WO-2010125831-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2010-11-04 WO disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS TRPM8, TRPM5, TRPM6 L3MBTL1 4792/4885MEN1 1593/4885KMT2A 941/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.