Pramiracetam

Pramiracetam

SCHEMBL120423

CC(C)N(CCNC(=O)CN1CCCC1=O)C(C)C.O=S(=O)(O)O

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Pramiracetam. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA1D known ✓ P25100 5/20 0.42
ADRA1A known ✓ P35348 5/20 0.42
ADRA1B known ✓ P35368 5/20 0.42
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.44
NQO2 P16083 1/20 0.44
TSHR P16473 2/20 0.42
KMT2A Q03164 2/20 0.42
ATAD2 Q6PL18 1/20 0.40
CECR2 Q9BXF3 1/20 0.40
PIK3CD O00329 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pramiracetam SCHEMBL195465 0.96 LMNA (0.48) LMNAHTTNQO2ADRA1DADRA1A
Pramiracetam SCHEMBL121209 0.95 LMNA (0.47) LMNAHTTNQO2ADRA1DADRA1A
Pramiracetam SCHEMBL11556360 0.95 LMNA (0.47) LMNAHTTNQO2ADRA1DADRA1A
Pramiracetam SCHEMBL1171471 0.94 LMNA (0.46) LMNAHTTNQO2ADRA1DADRA1A
Pramiracetam SCHEMBL4431064 0.85 LMNA (0.40) LMNAHTTNQO2ADRA1DADRA1A
Pramiracetam SCHEMBL2136275 0.84 LMNA (0.57) LMNAHTTNQO2ADRA1DADRA1A
Pramiracetam SCHEMBL9645954 0.82 LMNA (0.43) LMNAHTTNQO2ADRA1DADRA1A
SCHEMBL8961554 0.81 LMNA (0.45) LMNAHTTNQO2ADRA1DADRA1A
SCHEMBL11553497 0.81 HTT (0.50) LMNAHTTNQO2ADRA1DADRA1A
SCHEMBL11554851 0.81 TP53 (0.51) LMNAHTTNQO2ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 126 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104341333-B A kind of preparation method of pramiracetam sulfate BEIJING HUARUI DINGXIN TECHNOLOGY CO., LTD. (CN) 2016-03-02 CN claimed
CN-104341333-A Preparation method of Pramiracetam sulfate BEIJING HRDX MEDICINAL TECHNOLOGIES CO LTD 2015-02-11 CN claimed
US-20240247313-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2024-07-25 US disclosed
US-11905562-B2 Serotonin transporter gene and treatment of opioid-related disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2024-02-20 US disclosed
US-20210301346-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2021-09-30 US disclosed
US-20210290771-A1 ENGINEERED RECEPTOR/LIGAND SYSTEM FOR DELIVERY OF THERAPEUTIC AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2021-09-23 US disclosed
EP-3443955-B1 PHARMACEUTICAL COMPOSITIONS FOR IMPROVING MEMORY PERFORMANCE PHARNEXT (FR) 2021-06-16 EP disclosed
US-11000597-B2 Engineered receptor/ligand system for delivery of therapeutic agents UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2021-05-11 US disclosed
US-10995374-B2 Serotonin transporter gene and treatment of opioid-related disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2021-05-04 US disclosed
CN-111875530-A Pramipexole hydrate crystal and preparation method thereof 浙江朗华制药有限公司 2020-11-03 CN disclosed
EP-3692989-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS Afecta Pharmaceuticals, Inc. (US) 2020-08-12 EP disclosed
US-6323236-B2 PSYCHOLOGICAL DISORDERS UNIVERSITY OF CINCINNATI 2001-11-27 US disclosed
WO-2001074853-A2 METHODS AND PRODUCTS FOR REGULATING CELL MOTILITY MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-10-11 WO disclosed
US-20010023254-A1 Psychological disorders CINCINNATI, UNIVERSITY OF 2001-09-20 US disclosed
US-20010002404-A1 Fatty acid-pharmaceutical agent conjugates LUITPOLD PHARMACEUTICALS, INC. 2001-05-31 US disclosed
WO-2000050020-A2 USE OF SULFAMATE DERIVATIVES FOR TREATING IMPULSE CONTROL DISORDERS UNIVERSITY OF CINCINNATI (US) 2000-08-31 WO disclosed
WO-1999030690-A1 ORAL DELIVERY FORMULATION AXIA THERAPEUTICS, INC. (US) 1999-06-24 WO disclosed
US-5795909-A ANTICARCINOGENIC AND ANTITUMOR AGENTS; BREAST, COLON, OVARIANCANCERS NEUROMEDICA, INC. (US) 1998-08-18 US disclosed
WO-1991000085-A1 SUSTAINED RELEASE PHARMACEUTICAL COMPOSITIONS WARNER-LAMBERT COMPANY (US) 1991-01-10 WO disclosed
US-4973470-A COMPRESSED MIXTURE OF WATER SENSITIVE DRUG, CELLULOSE, AND LUBRICANT WARNER-LAMBERT COMPANY (US) 1990-11-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11905562-B2 Serotonin transporter gene and treatment of opioid-related disorders SLC6A4, SLC6A3, SLC6A2 ADRA1D 185/4885ADRA1A 300/4885ADRA1B 409/4885
US-20240247313-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS SLC6A4, SLC6A3, SLC6A2 ADRA1D 185/4885ADRA1A 300/4885ADRA1B 409/4885
US-20010002404-A1 Fatty acid-pharmaceutical agent conjugates FABP7, FFAR2, FFAR4 ADRA1D 1358/4885ADRA1A 775/4885ADRA1B 1354/4885
US-10995374-B2 Serotonin transporter gene and treatment of opioid-related disorders SLC6A4, SLC6A3, SLC6A2 ADRA1D 185/4885ADRA1A 300/4885ADRA1B 409/4885
US-20210301346-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS SLC6A4, SLC6A3, SLC6A2 ADRA1D 185/4885ADRA1A 300/4885ADRA1B 409/4885
US-20010023254-A1 Psychological disorders DRD2, DRD3, DRD1 ADRA1D 157/4885ADRA1A 387/4885ADRA1B 306/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.