SCHEMBL12200959

SCHEMBL12200959

COc1cccc(S(=O)(=O)Nc2cc(C)ccc2C(=O)O)c1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.61
CYP2C19 P33261 1/20 0.61
ACLY P53396 6/20 0.60
MCL1 Q07820 2/20 0.60
KEAP1 Q14145 2/20 0.57
NFE2L2 Q16236 2/20 0.57
FFAR4 Q5NUL3 1/20 0.57
METAP2 P50579 1/20 0.57
SLC16A3 O15427 1/20 0.53
AKR1C3 P42330 1/20 0.53
AKR1C2 P52895 1/20 0.53
PGR P06401 1/20 0.52
CYP1A2 P05177 1/20 0.52
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12201453 0.89 KEAP1 (0.56) CYP2C9CYP2C19ACLYMCL1KEAP1
SCHEMBL7316092 0.86 CYP2C9 (0.68) CYP2C9CYP2C19ACLYMCL1KEAP1
SCHEMBL23200342 0.86 MEN1 (0.66) KEAP1NFE2L2FFAR4METAP2SLC16A3
SCHEMBL23200290 0.84 CYP2C9 (0.76) CYP2C9CYP2C19ACLYMCL1FFAR4
SCHEMBL12201452 0.80 ACLY (0.74) CYP2C9CYP2C19ACLYMCL1METAP2
SCHEMBL12200777 0.80 FFAR4 (0.64) ACLYKEAP1NFE2L2FFAR4METAP2
SCHEMBL9402850 0.79 MCL1 (0.67) CYP2C9CYP2C19ACLYMCL1METAP2
SCHEMBL7318557 0.78 ACLY (0.54) CYP2C9CYP2C19ACLYMCL1METAP2
SCHEMBL9997061 0.78 MCL1 (0.67) MCL1KEAP1NFE2L2PGR
SCHEMBL3988508 0.78 METAP2 (0.74) CYP2C9MCL1KEAP1NFE2L2FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385820-B1 ANTHRANILIC ACID AMIDES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS ANTIARRHYTHMIA AGENTS, AND PHARMACEUTICAL PREPARATIONS THEREOF SANOFI AVENTIS DEUTSCHLAND (DE) 2011-10-12 EP disclosed
US-7332608-B2 Anthranilamides and methods of their use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-02-19 US disclosed
US-7332608-B2 Anthranilamides and methods of their use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-02-19 US disclosed
US-7235690-B2 Anthranilamides and methods of their use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-06-26 US disclosed
US-7235690-B2 Anthranilamides and methods of their use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-06-26 US disclosed
US-20070117807-A1 ANTHRANILAMIDES AND METHODS OF THEIR USE SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-05-24 US disclosed
US-20070117807-A1 ANTHRANILAMIDES AND METHODS OF THEIR USE SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070117807-A1 ANTHRANILAMIDES AND METHODS OF THEIR USE KCNH1, KCNH2, KCNJ2 CYP2C9 1109/4885CYP2C19 2213/4885ACLY 1447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.