SCHEMBL12366241

SCHEMBL12366241

[C-]#[N+]c1c(C(F)(F)F)cc(-c2ccccc2)n(Cc2cccc(C)c2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.42
TP53 P04637 6/20 0.41
MAPT P10636 5/20 0.41
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 2/20 0.37
HPGD P15428 2/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
ITGB7 P26010 1/20 0.36
ALDH1A1 P00352 5/20 0.36
CYP3A4 P08684 2/20 0.36
KDM4E B2RXH2 1/20 0.36
RECQL P46063 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366256 0.95 POLB (0.38) CNR1TP53MAPTMEN1KMT2A
SCHEMBL12366233 0.94 CNR1 (0.42) CNR1TP53MAPTMEN1KMT2A
SCHEMBL12366212 0.90 CNR1 (0.44) CNR1HPGDTSHRHSD17B10ITGB1
SCHEMBL12366295 0.90 ITGB1 (0.39) CNR1TP53MAPTHPGDTSHR
SCHEMBL12366245 0.89 CNR1 (0.43) CNR1TP53MAPTMEN1KMT2A
SCHEMBL12366286 0.89 MAPT (0.45) TP53MAPTPOLBALDH1A1KDM4E
SCHEMBL12366418 0.89 MAPT (0.42) TP53MAPTPOLBHPGDHSD17B10
SCHEMBL12366396 0.88 RXRA (0.41) CNR1TP53MAPTPOLBHPGD
SCHEMBL12366278 0.88 MAPT (0.45) TP53MAPTPOLBALDH1A1KDM4E
SCHEMBL12366740 0.88 PTGS2 (0.35) CNR1TP53MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed