SCHEMBL1241255

SCHEMBL1241255

Brc1ccc(CNC2CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
HRH3 Q9Y5N1 3/20 0.57
ACHE P22303 4/20 0.54
BCHE P06276 3/20 0.54
BACE1 P56817 3/20 0.54
POLB P06746 1/20 0.53
KDM1A O60341 1/20 0.50
HDAC1 Q13547 1/20 0.49
GRIN2B Q13224 1/20 0.48
MGAM O43451 1/20 0.44
SI P14410 1/20 0.44
ALDH1A1 P00352 1/20 0.44
PYCR1 P32322 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23124659 0.92 HRH3 (0.63) RAB9AMEN1KMT2AHRH3ACHE
SCHEMBL11431895 0.92 HRH3 (0.69) RAB9AMEN1KMT2AHRH3ACHE
SCHEMBL6224747 0.90 HRH3 (0.72) RAB9AMEN1KMT2AHRH3ACHE
SCHEMBL10073807 0.89 MEN1 (0.69) RAB9AMEN1KMT2AHRH3ACHE
SCHEMBL4139216 0.87 HRH3 (0.49) RAB9AMEN1KMT2AHRH3ACHE
SCHEMBL8806696 0.85 HRH3 (0.83) RAB9AMEN1KMT2AHRH3ACHE
SCHEMBL9460564 0.83 ACHE (0.48) RAB9AMEN1KMT2AHRH3ACHE
SCHEMBL8812297 0.81 HRH3 (0.60) HRH3ACHEBCHEBACE1POLB
SCHEMBL16055301 0.80 ACHE (0.52) MEN1KMT2AHRH3ACHEBCHE
SCHEMBL16538645 0.80 HRH3 (0.63) RAB9AMEN1KMT2AHRH3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116891454-B Small molecule inhibitor, preparation method and application thereof in preparation of anticancer drugs 山东省药学科学院 2025-05-16 CN disclosed
US-20250019371-A1 SMALL-MOLECULAR INHIBITORS FOR THE BETA-CATENIN/ B-CELL LYMPHOMA 9 PROTEIN-PROTEIN INTERACTION H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. 2025-01-16 US disclosed
US-20240391896-A1 SMALL MOLECULE COMPOUND TARGETING BCL9/BETA-CATENIN INTERACTION Nantong Jutai Biotech Co., Ltd. (CN) 2024-11-28 US disclosed
CN-118994095-A Small molecule inhibitor and preparation method and application thereof 上海医药工业研究院有限公司 2024-11-22 CN disclosed
CN-115151252-B Iron death inhibitor-diarylamine acetamides 维泰瑞隆有限公司 2024-08-27 CN disclosed
CN-117651697-A Small molecule compounds targeting BCL 9/beta-catenin interactions 南通聚太生物科技有限公司 2024-03-05 CN disclosed
CN-116891454-A Small molecule inhibitor, preparation method and application thereof in preparation of anticancer drugs 山东省药学科学院 2023-10-17 CN disclosed
US-20230159492-A1 FERROPTOSIS INHIBITORS - DIARYLAMINE PARA-ACETAMIDES Sironax Ltd. (KY) 2023-05-25 US disclosed
US-20230159492-A1 FERROPTOSIS INHIBITORS - DIARYLAMINE PARA-ACETAMIDES Sironax Ltd. (KY) 2023-05-25 US disclosed
WO-2023077057-A1 SMALL-MOLECULAR INHIBITORS FOR THE BETA-CATENIN/ B-CELL LYMPHOMA 9 PROTEIN-PROTEIN INTERACTION H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2023-05-04 WO disclosed
WO-2021055936-A1 SMALL-MOLECULE INHIBITORS FOR THE Β-CATENIN/B-CELL LYMPHOMA 9 PROTEIN−PROTEIN INTERACTION H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2021-03-25 WO disclosed
WO-2021055936-A1 SMALL-MOLECULE INHIBITORS FOR THE Β-CATENIN/B-CELL LYMPHOMA 9 PROTEIN−PROTEIN INTERACTION H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2021-03-25 WO disclosed
CN-111646978-A N2-substituted alkoxy aromatic ring-2-aminopyrimidine derivatives and application thereof 浙江大学 2020-09-11 CN disclosed
US-10407422-B2 Triazolopyridine inhibitors of myeloperoxidase BRISTOL-MYERS SQUIBB COMPANY (US) 2019-09-10 US disclosed
US-20190023701-A1 TRIAZOLOPYRIDINE INHIBITORS OF MYELOPEROXIDASE BRISTOL MYERS SQUIBB CO (US) 2019-01-24 US disclosed
WO-2017040449-A1 TRIAZOLOPYRIDINE INHIBITORS OF MYELOPEROXIDASE BRISTOL-MYERS SQUIBB COMPANY (US) 2017-03-09 WO disclosed
WO-2017040449-A1 TRIAZOLOPYRIDINE INHIBITORS OF MYELOPEROXIDASE BRISTOL-MYERS SQUIBB COMPANY (US) 2017-03-09 WO disclosed
US-7879808-B2 potent activity against resistant pneumococci; for treating domestic fowl MEIJI SEIKA KAISHA, LTD. (JP) 2011-02-01 US disclosed
US-20100210570-A1 LINCOMYCIN DERIVATIVES AND ANTIMICROBIAL AGENTS COMPRISING THE SAME AS ACTIVE INGREDIENT MEIJI SEIKA KAISHA LTD. (JP) 2010-08-19 US disclosed
EP-2151447-A1 LINCOMYCIN DERIVATIVES AND ANTIBACTERIAL AGENTS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Meiji Seika Kaisha Ltd. (JP) 2010-02-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240391896-A1 SMALL MOLECULE COMPOUND TARGETING BCL9/BETA-CATENIN INTERACTION BCL9, BCL9L, BCL2L11 RAB9A 48/4885MEN1 2556/4885KMT2A 3657/4885
US-20190023701-A1 TRIAZOLOPYRIDINE INHIBITORS OF MYELOPEROXIDASE EPX, MPO, SERPINB1 RAB9A 3993/4885MEN1 4641/4885KMT2A 2066/4885
US-10407422-B2 Triazolopyridine inhibitors of myeloperoxidase EPX, MPO, SERPINB1 RAB9A 3993/4885MEN1 4641/4885KMT2A 2066/4885
US-20100210570-A1 LINCOMYCIN DERIVATIVES AND ANTIMICROBIAL AGENTS COMPRISING THE SAME AS ACTIVE INGREDIENT LAS1L, LCLAT1, LYPLA1 RAB9A 828/4885MEN1 977/4885KMT2A 3710/4885
US-20250019371-A1 SMALL-MOLECULAR INHIBITORS FOR THE BETA-CATENIN/ B-CELL LYMPHOMA 9 PROTEIN-PROTEIN INTERACTION BCL9, BCL9L, BCL6 RAB9A 455/4885MEN1 3726/4885KMT2A 3118/4885
US-20230159492-A1 FERROPTOSIS INHIBITORS - DIARYLAMINE PARA-ACETAMIDES AIFM2, FECH, GPX4 RAB9A 2759/4885MEN1 2123/4885KMT2A 2622/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.