SCHEMBL12467259

SCHEMBL12467259

CCc1cc(Cl)cc2c1OCO2

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
CYP3A4 P08684 2/20 0.39
NQO2 P16083 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
LTC4S Q16873 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAOB P27338 2/20 0.33
POLB P06746 2/20 0.33
AHR P35869 1/20 0.33
MAPT P10636 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
AOC3 Q16853 1/20 0.33
ACVRL1 P37023 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13186975 0.87 MTNR1A (0.36) TAAR1MAOB
SCHEMBL25844870 0.82 MAOB (0.34) ALDH1A1CYP3A4LTC4SSMN1; SMN2MAOB
SCHEMBL25845153 0.81 ALOX5 (0.36) ALDH1A1CYP3A4LTC4SMAOBPOLB
SCHEMBL5271445 0.80 ALDH1A1 (0.35) ALDH1A1CYP3A4LTC4SSMN1; SMN2MAOB
SCHEMBL11081166 0.79 AHR (0.47) ALDH1A1CYP3A4SMN1; SMN2MAOBAHR
SCHEMBL6542530 0.77 CYP3A4 (0.39) ALDH1A1CYP3A4NQO2SMN1; SMN2MAOB
SCHEMBL12484333 0.76 NPC1 (0.37) ALDH1A1CYP3A4NQO2SMN1; SMN2POLB
SCHEMBL14337789 0.75 DHFR (0.49) ALDH1A1CYP3A4SMN1; SMN2MAOBPOLB
SCHEMBL9921215 0.74 CYP3A4 (0.37) ALDH1A1CYP3A4MAOB
SCHEMBL10044946 0.74 ALDH1A1 (0.47) ALDH1A1CYP3A4SMN1; SMN2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170216283-A1 COMPOUNDS AND USES ASTRAZENECA AB (SE) 2017-08-03 US disclosed
US-20170216283-A1 COMPOUNDS AND USES ASTRAZENECA AB (SE) 2017-08-03 US disclosed
US-9657001-B2 Compounds and uses ASTRAZENECA AB (SE) 2017-05-23 US disclosed
US-9657001-B2 Compounds and uses ASTRAZENECA AB (SE) 2017-05-23 US disclosed
US-20160326143-A1 COMPOUNDS AND USES ASTRAZENECA AB (SE) 2016-11-10 US disclosed
US-20160326143-A1 COMPOUNDS AND USES ASTRAZENECA AB (SE) 2016-11-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170216283-A1 COMPOUNDS AND USES LTC4S, LTB4R2, LTA4H ALDH1A1 268/4885CYP3A4 215/4885NQO2 279/4885
US-20160326143-A1 COMPOUNDS AND USES LTC4S, LTB4R2, LTA4H ALDH1A1 268/4885CYP3A4 215/4885NQO2 279/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.