SCHEMBL12633801

SCHEMBL12633801

COc1cc2c(cc1OC)C(C)N(C)C(C)C2

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.55
SMN1; SMN2 Q16637 1/20 0.47
CA7 P43166 1/20 0.46
BRD4 O60885 2/20 0.44
TSHR P16473 1/20 0.42
RAD52 P43351 1/20 0.42
HTR1A P08908 1/20 0.42
PDE4B Q07343 1/20 0.41
PDE4D Q08499 1/20 0.41
KCNN2 Q9H2S1 3/20 0.41
KCNN3 Q9UGI6 3/20 0.41
KCNN1 Q92952 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26956140 0.87 HTR2C (0.47) MAOASMN1; SMN2CA7HTR1AMAPT
SCHEMBL29516257 0.87 MAOA (0.43) MAOASMN1; SMN2CA7BRD4TSHR
SCHEMBL29516230 0.81 SIRT6 (0.43) MAOASMN1; SMN2CA7MAPT
SCHEMBL26956142 0.77 OPRM1 (0.49) TSHR
Argemonine SCHEMBL3865650 0.77 HTR1A (0.58) MAOARAD52HTR1ACYP3A4
Argemonine SCHEMBL30435899 0.77 HTR1A (0.58) MAOARAD52HTR1ACYP3A4
SCHEMBL3159301 0.74 ACHE (0.56) MAOATSHRRAD52CYP3A4MAPT
SCHEMBL4565692 0.74 ACHE (0.56) MAOATSHRRAD52CYP3A4MAPT
SCHEMBL1760713 0.72 MAOA (0.97) MAOASMN1; SMN2CA7BRD4RAD52
SCHEMBL29382740 0.72 MAOA (0.97) MAOASMN1; SMN2CA7BRD4RAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075957-A1 TETRAHYDROISOQUINOLINE COMPOUNDS, PREPARATION METHODS AND USES THEREOF 沈阳药科大学 (CN) 2011-06-30 WO disclosed