SCHEMBL1264341

SCHEMBL1264341

Brc1ccc2c(c1)CCNCC2

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 3/20 0.77
ASIC3 Q9UHC3 1/20 0.77
HTR2C P28335 7/20 0.57
HTR2B P41595 6/20 0.57
HTR2A P28223 4/20 0.57
MELK Q14680 1/20 0.53
PARP10 Q53GL7 2/20 0.48
PARP11 Q9NR21 1/20 0.48
PARP1 P09874 1/20 0.48
ADCY6 O43306 1/20 0.48
ADCY3 O60266 1/20 0.48
ADCY9 O60503 1/20 0.48
ADCY5 O95622 1/20 0.48
ADCY8 P40145 1/20 0.48
ADCY7 P51828 1/20 0.48
ADCY2 Q08462 1/20 0.48
ADCY1 Q08828 1/20 0.48
ADCY4 Q8NFM4 1/20 0.48
DRD2 P14416 1/20 0.47
DRD1 P21728 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL21753269 0.98 PNMT (0.74) PNMTASIC3HTR2CHTR2BHTR2A
SCHEMBL12895998 0.92 PNMT (0.67) PNMTASIC3HTR2CHTR2BHTR2A
SCHEMBL29473102 0.87 PNMT (1.00) PNMTASIC3HTR2CHTR2BHTR2A
SCHEMBL505055 0.87 ASIC3 (1.00) PNMTASIC3HTR2CHTR2BHTR2A
SCHEMBL552932 0.87 PNMT (1.00) PNMTASIC3HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL1017313 0.85 ASIC3 (0.96) PNMTASIC3HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL1266299 0.85 PNMT (0.96) PNMTASIC3HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL29528420 0.85 PNMT (0.96) PNMTASIC3HTR2CHTR2BHTR2A
SCHEMBL13594 0.83
Ammonia Solution, Strong SCHEMBL8701960 0.80 PNMT (0.56) PNMTASIC3PARP10PARP11PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 108 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4547246-A2 COMPOUNDS AS INHIBITORS OF AXL Arcus Biosciences, Inc. (US) 2025-05-07 EP disclosed
US-12195482-B1 Compounds as inhibitors of AXL ARCUS BIOSCIENCES, INC. (US) 2025-01-14 US disclosed
US-20240425526-A1 COMPOUNDS AS INHIBITORS OF AXL ARCUS BIOSCIENCES, INC. (US) 2024-12-26 US disclosed
EP-3601229-B1 TETRAHYDRO-BENZO[D]AZEPINE DERIVATIVES AS GPR120 MODULATORS CALDAN THERAPEUTICS LTD (GB) 2024-11-06 EP disclosed
CN-115594669-B Parallel ring derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2024-11-05 CN disclosed
US-20240226115-A1 AXL INHIBITOR COMPOUNDS ARCUS BIOSCIENCES, INC. 2024-07-11 US disclosed
US-20240226115-A1 AXL INHIBITOR COMPOUNDS ARCUS BIOSCIENCES, INC. 2024-07-11 US disclosed
US-20240174631-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR MODULATING FGF ACTIVITY RECOVERY THERAPEUTICS, INC. 2024-05-30 US disclosed
WO-2024006726-A2 COMPOUNDS AS INHIBITORS OF AXL ARCUS BIOSCIENCES, INC. (US) 2024-01-04 WO disclosed
US-20230416277-A1 COMPOUNDS AS INHIBITORS OF AXL ARCUS BIOSCIENCES, INC. 2023-12-28 US disclosed
US-20080113967-A1 ENZYME MODULATORS AND TREATMENTS DECIPHERA PHARMACEUTICALS, LLC (US) 2008-05-15 US disclosed
US-20080113967-A1 ENZYME MODULATORS AND TREATMENTS DECIPHERA PHARMACEUTICALS, LLC (US) 2008-05-15 US disclosed
US-7304050-B2 Antibacterial agents PFIZER INC. (US) 2007-12-04 US disclosed
US-7304050-B2 Antibacterial agents PFIZER INC. (US) 2007-12-04 US disclosed
US-20070078121-A1 Enzyme modulators and treatments DECIPHERA PHARMACEUTICALS, LLC 2007-04-05 US disclosed
US-20070078121-A1 Enzyme modulators and treatments DECIPHERA PHARMACEUTICALS, LLC 2007-04-05 US disclosed
EP-1594494-A1 OXAZOLIDINONE DERIVATIVES N-SUBSTITUTED BY A BICYCLIC RING, FOR USE AS ANTIBACTERIAL AGENTS Warner-Lambert Company LLC (US) 2005-11-16 EP disclosed
US-20040224939-A1 Antibacterial agents CHUPAK LOUIS S (US) 2004-11-11 US disclosed
WO-2004069244-A1 OXAZOLIDINONE DERIVATIVES N-SUBSTITUTED BY A BICYCLIC RING, FOR USE AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2004-08-19 WO disclosed
EP-1011679-B1 USE OF 8-NITRO-2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINES FOR THE MANUFACTURE OF A PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF SLEEP DISORDERS ADDEX PHARMACEUTICALS SA (CH) 2003-07-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040224939-A1 Antibacterial agents MRPL21, RPN2, FBL PNMT 3757/4885ASIC3 4530/4885HTR2C 4790/4885
US-12195482-B1 Compounds as inhibitors of AXL AXL, FLT3, BTK PNMT 3497/4885ASIC3 2252/4885HTR2C 4165/4885
US-20240174631-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR MODULATING FGF ACTIVITY FGF1, FGF2, FGFR1 PNMT 4852/4885ASIC3 544/4885HTR2C 1517/4885
US-20240226115-A1 AXL INHIBITOR COMPOUNDS AXL, BTK, MERTK PNMT 3997/4885ASIC3 2819/4885HTR2C 4367/4885
US-20070078121-A1 Enzyme modulators and treatments ABL1, ABL2, LCK PNMT 998/4885ASIC3 4164/4885HTR2C 2813/4885
US-20240425526-A1 COMPOUNDS AS INHIBITORS OF AXL AXL, FLT3, BTK PNMT 3497/4885ASIC3 2252/4885HTR2C 4165/4885
US-20080113967-A1 ENZYME MODULATORS AND TREATMENTS ABL2, BRAF, MAP3K1 PNMT 1190/4885ASIC3 4447/4885HTR2C 3311/4885
US-20230416277-A1 COMPOUNDS AS INHIBITORS OF AXL AXL, FLT3, BTK PNMT 3497/4885ASIC3 2252/4885HTR2C 4165/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.