SCHEMBL12840913

SCHEMBL12840913

C=CC(=O)N1CCN(c2ccc(N)c(OC)c2)CC1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 1/20 0.48
ACHE P22303 6/20 0.46
EGFR P00533 4/20 0.45
ALDH1A1 P00352 1/20 0.44
CCR1 P32246 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13362096 0.85 HTR1A (0.51) ALDH1A1CCR1
SCHEMBL11294977 0.85 CCR1 (0.46) ALDH1A1CCR1
SCHEMBL2205957 0.85 CASP6 (0.59)
SCHEMBL4174848 0.84 L3MBTL1 (0.61) ALDH1A1CCR1
SCHEMBL15358736 0.83 ALDH1A1 (0.53) ALDH1A1
SCHEMBL4170621 0.82 MAPT (0.47) ALDH1A1CCR1
SCHEMBL2723108 0.82 ALK (0.53) ALDH1A1CCR1
SCHEMBL4171024 0.82 CCR1 (0.51) ALDH1A1CCR1
SCHEMBL13178104 0.82 SIRT6 (0.52) CCR1
SCHEMBL4172479 0.82 ALK (0.50) ALDH1A1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478539-B Novel DCLK1 inhibitor and preparation method and application thereof 中国人民解放军海军军医大学 2024-02-02 CN disclosed
CN-114478539-A Novel DCLK1 inhibitor and preparation method and application thereof 中国人民解放军海军军医大学 2022-05-13 CN disclosed
WO-2011034907-A2 PROTEIN KINASE CONJUGATES AND INHIBITORS AVILA THERAPEUTICS, INC. (US) 2011-03-24 WO disclosed