SCHEMBL4172479

SCHEMBL4172479

COc1cc(N2CCN(C(=O)C(C)(C)C)CC2)ccc1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.50
TP53 P04637 1/20 0.49
PDK2 Q15119 1/20 0.46
LMNA P02545 3/20 0.44
HTT P42858 2/20 0.44
MAPT P10636 2/20 0.44
ALOX15 P16050 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 1/20 0.44
CCR1 P32246 2/20 0.43
TSHR P16473 2/20 0.42
NPC1 O15118 1/20 0.42
TYR P14679 1/20 0.41
CASP6 P55212 1/20 0.41
GFER P55789 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4162968 0.88 LMNA (0.46) ALKTP53LMNAHTTMAPT
SCHEMBL18997523 0.85 ALK (0.51) ALKTP53PDK2LMNAHTT
SCHEMBL19002642 0.85 ACHE (0.52) ALKTP53PDK2LMNAHTT
SCHEMBL11294977 0.85 CCR1 (0.46) LMNAHTTMAPTALOX15L3MBTL1
SCHEMBL2205957 0.85 CASP6 (0.59) ALKLMNAMAPTCASP6GFER
SCHEMBL13362096 0.85 HTR1A (0.51) LMNAHTTMAPTALOX15L3MBTL1
SCHEMBL1707770 0.85 MAPT (0.57) ALKPDK2LMNAMAPTALDH1A1
SCHEMBL4177069 0.84 EGFR (0.46) ALKTP53PDK2LMNAHTT
SCHEMBL4174848 0.84 L3MBTL1 (0.61) ALKPDK2HTTMAPTL3MBTL1
SCHEMBL4172363 0.84 MAPT (0.45) ALKTP53LMNAMAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061299-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF AVILA THERAPEUTICS, INC. (US) 2012-05-10 WO disclosed