SCHEMBL12846266

SCHEMBL12846266

Cc1cc(C2=NOC(c3cc(Cl)cc(Cl)c3)(C(F)(F)F)C2)ccc1C(=O)NCC(=O)N(C)C

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.38
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
P2RX7 Q99572 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ELOVL6 Q9H5J4 1/20 0.31
CYP3A4 P08684 1/20 0.30
KMT2A Q03164 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL737408 0.91 EGLN1 (0.36) CA1CA2KDM4ELMNAL3MBTL1
SCHEMBL740369 0.90 CA1 (0.34) CA1CA2P2RX7KDM4ELMNA
SCHEMBL30233680 0.90 CASP1 (0.39) KDM4ELMNAL3MBTL1SMN1; SMN2
SCHEMBL739739 0.90 EGLN1 (0.36) CA1CA2KDM4ELMNACYP3A4
SCHEMBL12846265 0.90 HDAC4 (0.38) HDAC4CA1CA2KDM4EELOVL6
SCHEMBL738538 0.90 CYP3A4 (0.38) CA1CA2ELOVL6CYP3A4KMT2A
SCHEMBL15059546 0.89 TTK (0.36) HDAC4CA1CA2LMNAELOVL6
SCHEMBL15059547 0.89 TTK (0.36) HDAC4CA1CA2LMNAELOVL6
SCHEMBL12846262 0.88 TTK (0.33) HDAC4CA1CA2KDM4EELOVL6
SCHEMBL119374 0.88 PTGES (0.35) CA1CA2KDM4ELMNAELOVL6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240239759-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS INTERVET INC. (US) 2024-07-18 US disclosed
EP-3473101-B1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS FOR FELINES INTERVET INT BV (NL) 2021-05-12 EP disclosed
US-20210061775-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS INTERVET INC. (US) 2021-03-04 US disclosed
EP-3473101-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS FOR FELINES Intervet International B.V. (NL) 2019-04-24 EP disclosed
US-20180155301-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS INTERVET INC. (US) 2018-06-07 US disclosed
US-20160332975-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS INTERVET INC. (US) 2016-11-17 US disclosed
US-20150111936-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS INTERVET INC (US) 2015-04-23 US disclosed
EP-2545777-A1 Isoxazoline compositions and their use as antiparasitics Intervet International B.V. (NL) 2013-01-16 EP disclosed
US-20110059988-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS INTERVET INTERNATIONAL B.V. 2011-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160332975-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS PRDX5, TUBA3C, TUBA1C HDAC4 504/4885CA1 1771/4885CA2 651/4885
US-20210061775-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS PRDX5, TUBA3C, TUBA1C HDAC4 504/4885CA1 1771/4885CA2 651/4885
US-20180155301-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS PRDX5, TUBA3C, TUBA1C HDAC4 504/4885CA1 1771/4885CA2 651/4885
US-20150111936-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS PRDX5, TUBA3C, EPX HDAC4 459/4885CA1 1649/4885CA2 595/4885
US-20240239759-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS PRDX5, TUBA3C, TUBA1C HDAC4 504/4885CA1 1771/4885CA2 651/4885
US-20110059988-A1 ISOXAZOLINE COMPOSITIONS AND THEIR USE AS ANTIPARASITICS PRDX5, TUBA3C, AADAC HDAC4 411/4885CA1 1922/4885CA2 661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.