SCHEMBL13045

SCHEMBL13045

Cc1cccc(-c2cccnc2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.62
CYP3A4 P08684 2/20 0.62
ALDH1A1 P00352 1/20 0.62
CYP1A2 P05177 1/20 0.62
NPY5R Q15761 1/20 0.61
MKNK1 Q9BUB5 2/20 0.60
MKNK2 Q9HBH9 2/20 0.60
MEN1 O00255 1/20 0.60
PSIP1 O75475 1/20 0.60
AXL P30530 1/20 0.60
GABRG2 P18507 1/20 0.55
GABRB3 P28472 1/20 0.55
GABRA3 P34903 1/20 0.55
EPHX2 P34913 1/20 0.54
PRMT6 Q96LA8 1/20 0.54
CYP17A1 P05093 2/20 0.53
CYP19A1 P11511 2/20 0.53
CYP11B1 P15538 2/20 0.53
CYP11B2 P19099 2/20 0.53
KMO O15229 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12373158 0.96 NPY5R (0.58) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL21982139 0.96 NPY5R (0.58) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL19009230 0.96 NPY5R (0.58) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL19309598 0.94 NPY5R (0.56) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL22693745 0.90 CYP2A6 (0.60) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL18960598 0.89 NPY5R (0.52) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL13624039 0.86 CYP2A6 (0.56) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL18267891 0.86 CYP19A1 (0.67) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL10262832 0.85 CYP2A6 (0.65) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R
SCHEMBL12070458 0.85 CYP2A6 (0.65) CYP2A6CYP3A4ALDH1A1CYP1A2NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 403 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663204-B1 C-KIT MODULATORS AND METHODS OF USE EXELIXIS INC (US) 2014-05-07 EP claimed
US-20080096892-A1 C-Kit Modulators And Methods Of Use EXELIXIS, INC. (US) 2008-04-24 US claimed
US-20240244946-A1 ORGANIC LIGHT EMITTING DIODE COMPRISING ORGANOMETALLIC COMPOUND AND PLURALITY OF HOST MATERIALS LG DISPLAY CO., LTD. (KR) 2024-07-18 US disclosed
WO-2024145931-A1 SMALL MOLECULE INHIBITOR FOR β-CATENIN/BCL9 PROTEIN-PROTEIN INTERACTION AND USE THEREOF 上海医药工业研究院有限公司 2024-07-11 WO disclosed
US-11877506-B2 Polycyclic aromatic compound KWANSEI GAKUIN EDUCATIONAL FOUNDATION (JP) 2024-01-16 US disclosed
EP-3935129-B1 LIGANDS FOR NANO-SIZED MATERIALS MERCK PATENT GMBH (DE) 2023-11-29 EP disclosed
US-11832513-B2 Materials for electronic devices MERCK PATENT GMBH (DE) 2023-11-28 US disclosed
US-11832513-B2 Materials for electronic devices MERCK PATENT GMBH (DE) 2023-11-28 US disclosed
US-20230373941-A1 COMPOUNDS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2023-11-23 US disclosed
US-20230373941-A1 COMPOUNDS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2023-11-23 US disclosed
US-20230371358-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-11-16 US disclosed
US-20050148623-A1 Prevent reproduct of aids virus ABBVIE INC. 2005-07-07 US disclosed
WO-2004069158-A2 SUBSTITUTED PYRAZOLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO., INC. (US) 2004-08-19 WO disclosed
US-4937346-A Phenyl-azacykloalkanes Carlsson, Per Arvid Emil (SE) 1990-06-26 US disclosed
US-4719219-A Phenyl-azacycloalkanes and use thereof in treatment of central nervous system disorders Carlsson, Per A. E. (SE) 1988-01-12 US disclosed
US-4426386-A CNS DISORDERS ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1984-01-17 US disclosed
EP-0084920-A2 New compounds useful as intermediates or starting materials for preparation of therapeutically useful phenyl-azacycloalkanes Carlsson, Per Arvid Emil (SE) 1983-08-03 EP disclosed
EP-0030526-A1 New phenyl-azacycloalkanes, processes for preparation and pharmaceutical preparations for such compounds Astra Läkemedel Aktiebolag (SE) 1981-06-17 EP disclosed
WO-1981001552-A1 NEW PHENYL-AZACYCLOALKANES ASTRA LAEKEMEDEL AB (SE) 1981-06-11 WO disclosed
US-4128651-A Bis-quaternary pyridinium-2-aldoxime salts and a process for their preparation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1978-12-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080096892-A1 C-Kit Modulators And Methods Of Use KIT, PRKCH, PRKCB CYP2A6 4760/4885CYP3A4 4747/4885ALDH1A1 2190/4885
US-11877506-B2 Polycyclic aromatic compound F11, C1R, RNF31 CYP2A6 1085/4885CYP3A4 685/4885ALDH1A1 2814/4885
US-11832513-B2 Materials for electronic devices PNMT, DDT, COMT CYP2A6 120/4885CYP3A4 35/4885ALDH1A1 321/4885
US-20050148623-A1 Prevent reproduct of aids virus SERPINB1, PRSS1, SERPINA3 CYP2A6 580/4885CYP3A4 481/4885ALDH1A1 1209/4885
US-20240244946-A1 ORGANIC LIGHT EMITTING DIODE COMPRISING ORGANOMETALLIC COMPOUND AND PLURALITY OF HOST MATERIALS GPX1, PER2, SOD1 CYP2A6 2160/4885CYP3A4 1109/4885ALDH1A1 10/4885
US-20230373941-A1 COMPOUNDS FOR ELECTRONIC DEVICES CYP2E1, GPX1, ERCC1 CYP2A6 188/4885CYP3A4 114/4885ALDH1A1 115/4885
US-20230371358-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES LIFR, SOD1, ROS1 CYP2A6 4425/4885CYP3A4 2401/4885ALDH1A1 569/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.