Epigalocatechin Gallate

Epigalocatechin Gallate

SCHEMBL13624466

O=C(O[C@@H]1Cc2c(O)cc(O)cc2OC1c1cc(O)c(O)c(O)c1)c1cc(O)c(O)c(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 10/20 1.00
BACE1 P56817 5/20 1.00
MMP2 P08253 5/20 1.00
MMP7 P09237 5/20 1.00
MMP14 P50281 5/20 1.00
BCL2 P10415 4/20 1.00
PSMB5 P28074 4/20 1.00
SNCA P37840 4/20 1.00
PGD P52209 4/20 1.00
MET P08581 3/20 1.00
KDM4E B2RXH2 3/20 1.00
MEN1 O00255 3/20 1.00
MAPT P10636 3/20 1.00
RECQL P46063 3/20 1.00
KMT2A Q03164 3/20 1.00
TDP1 Q9NUW8 3/20 1.00
PKM P14618 3/20 1.00
PKMYT1 Q99640 2/20 1.00
PGAM1 P18669 2/20 1.00
SIRT6 Q8N6T7 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Epigalocatechin Gallate SCHEMBL29389587 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Gallocatechin Gallate SCHEMBL30977114 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Epigalocatechin Gallate SCHEMBL30014282 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Epigalocatechin Gallate SCHEMBL30909383 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Epigalocatechin Gallate SCHEMBL10198783 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Epigalocatechin Gallate SCHEMBL14423426 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Epigalocatechin Gallate SCHEMBL35258 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Gallocatechin Gallate SCHEMBL49461 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Epigalocatechin Gallate SCHEMBL8426376 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14
Epigalocatechin Gallate SCHEMBL29410018 1.00 DYRK1A (1.00) DYRK1ABACE1MMP2MMP7MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11744820-B2 Inhibitors of microbially induced amyloid AXIAL THERAPEUTICS, INC. (US) 2023-09-05 US disclosed
US-20210252097-A1 POLYPHARMACEUTICAL DRUG COMPOSITIONS AND RELATED METHODS AVETA BIOMICS, INC. (US) 2021-08-19 US disclosed
EP-3560587-A1 METHOD FOR SYNTHESIS OF A METAL ORGANIC FRAMEWORK COMPOSITE Ecole Polytechnique Fédérale de Lausanne (EPFL) (CH) 2019-10-30 EP disclosed
US-9795597-B2 Cyclopropylamines as LSD1 inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2017-10-24 US disclosed
US-9408407-B2 Compounds, compositions, and methods for reducing or eliminating bitter taste CHROMOCELL CORPORATION (US) 2016-08-09 US disclosed
US-20160220547-A1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2016-08-04 US disclosed
US-20150313906-A1 COMBINATION GLAXOSMITHKLINE LLC 2015-11-05 US disclosed
US-20150313906-A1 COMBINATION GLAXOSMITHKLINE LLC 2015-11-05 US disclosed
US-20150306099-A1 COMBINATION GLAXOSMITHKLINE LLC 2015-10-29 US disclosed
US-20150306099-A1 COMBINATION GLAXOSMITHKLINE LLC 2015-10-29 US disclosed
US-20150237900-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR REDUCING OR ELIMINATING BITTER TASTE CHROMOCELL CORP (US) 2015-08-27 US disclosed
US-8865779-B2 Compounds, compositions, and methods for reducing or eliminating bitter taste CHROMOCELL CORPORATION (US) 2014-10-21 US disclosed
US-20130287918-A1 MICROBICIDAL COMPOSITION DUPONT NUTRITION DIOSCIENCES APS (DK) 2013-10-31 US disclosed
US-20130287918-A1 MICROBICIDAL COMPOSITION DUPONT NUTRITION DIOSCIENCES APS (DK) 2013-10-31 US disclosed
US-20130096209-A1 Compounds, Compositions, And Methods For Reducing Or Eliminating Bitter Taste KRAFT FOODS GLOBAL BRANDS LLC (US) 2013-04-18 US disclosed
EP-2119712-A1 NOVEL METHYLATED CATECHIN AND COMPOSITION CONTAINING THE SAME Incorporated Administrative Agency National Agriculture and Food Research Organization (JP) 2009-11-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160220547-A1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS KDM1B, KDM1A, KDM3B DYRK1A 1348/4885BACE1 1181/4885MMP2 3081/4885
US-20210252097-A1 POLYPHARMACEUTICAL DRUG COMPOSITIONS AND RELATED METHODS PCBP1, CYP3A5, ABCB1 DYRK1A 2796/4885BACE1 1152/4885MMP2 4763/4885
US-20150306099-A1 COMBINATION VHL, CA5A, HRAS DYRK1A 2340/4885BACE1 3057/4885MMP2 4608/4885
US-11744820-B2 Inhibitors of microbially induced amyloid APP, PSEN1, BACE1 DYRK1A 4091/4885BACE1 3/4885MMP2 1057/4885
US-20150237900-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR REDUCING OR ELIMINATING BITTER TASTE TAS2R5, TAS2R20, TAS2R10 DYRK1A 3989/4885BACE1 4010/4885MMP2 4785/4885
US-20150313906-A1 COMBINATION EZH2, BMI1, DOT1L DYRK1A 583/4885BACE1 2450/4885MMP2 4137/4885
US-20130096209-A1 Compounds, Compositions, And Methods For Reducing Or Eliminating Bitter Taste TAS2R5, TAS2R20, TAS2R10 DYRK1A 3989/4885BACE1 4010/4885MMP2 4785/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.