SCHEMBL13626525

SCHEMBL13626525

Cc1cccc2c1CC(C(=O)Nc1ccc(C(=N)N3CCCC3)cc1)N(C(=O)Nc1ccc(Cl)cc1)C2

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CFTR P13569 7/20 0.45
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.40
PKM P14618 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
RHOA P61586 1/20 0.40
MAPT P10636 1/20 0.39
P2RX7 Q99572 1/20 0.39
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
UBE2M P61081 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626492 0.87 CFTR (0.55) CFTRMEN1GAAKMT2ALMNA
SCHEMBL13626527 0.86 CFTR (0.46) CFTRMEN1GAAKMT2ALMNA
SCHEMBL13626533 0.81 SMN1; SMN2 (0.49) CFTRMAPTL3MBTL1ALDH1A1TSHR
SCHEMBL13626502 0.78 LMNA (0.58) CFTRMEN1GAAKMT2ALMNA
SCHEMBL13626522 0.78 CFTR (0.40) CFTRMEN1GAAKMT2ATAS1R3
SCHEMBL13626503 0.73 CFTR (0.56) CFTRMEN1GAAKMT2ALMNA
SCHEMBL13626514 0.69 LMNA (0.53) CFTRMEN1GAAKMT2ALMNA
SCHEMBL13626515 0.69 LMNA (0.53) CFTRMEN1GAAKMT2ALMNA
SCHEMBL12134196 0.69 F10 (0.57) MEN1KMT2ALMNARAB9A
SCHEMBL13626504 0.68 NAMPT (0.51) CFTRMEN1GAAKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612089-B2 Tetrahydroisoquinolines as factor Xa inhibitors PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-03 US disclosed
US-7612089-B2 Tetrahydroisoquinolines as factor Xa inhibitors PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-03 US disclosed