SCHEMBL1363051

SCHEMBL1363051

CC1(C)OB(c2cccc(CN3CCN(C(=O)O)[C@@](C)(C(C)(C)C)C3)c2)OC1(C)C

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LIPG Q9Y5X9 2/20 0.41
LPL P06858 1/20 0.41
KDM4E B2RXH2 5/20 0.34
ALDH1A1 P00352 4/20 0.34
MAPK1 P28482 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ROCK1 Q13464 1/20 0.34
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HIF1A Q16665 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
FAAH O00519 2/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1632683 0.83 KDM4E (0.48) KDM4EALDH1A1MAPK1SMN1; SMN2NPSR1
SCHEMBL3045151 0.81 LIPG (0.47) LIPGLPLKDM4EALDH1A1MAPK1
SCHEMBL1362390 0.78 FAAH (0.41) KDM4EALDH1A1FAAHLMNAMAPT
SCHEMBL25425656 0.77 LIPG (0.40) LIPGLPLKDM4EALDH1A1MAPK1
SCHEMBL1363050 0.76 LIPG (0.39) LIPGLPLKDM4EALDH1A1NPSR1
SCHEMBL3399375 0.76 LIPG (0.42) LIPGLPLMEN1KMT2A
SCHEMBL3041956 0.76 GLS (0.47) LIPGLPLALDH1A1PRMT5WDR77
SCHEMBL29964482 0.76 GLS (0.47) LIPGLPLALDH1A1PRMT5WDR77
SCHEMBL3399142 0.76 LIPG (0.42) LIPGLPLMEN1KMT2A
SCHEMBL1631726 0.75 CYP2E1 (0.40) KDM4EALDH1A1CYP2C9FAAHLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067408-B2 Dual pharmacophores—PDE4-muscarinic antagonistics GLAXO GROUP LIMITED (GB) 2011-11-29 US disclosed