SCHEMBL13634625

SCHEMBL13634625

O=C(Nc1ccccc1C(=O)NC1CCOCC1)c1coc(N2CC[C@@H](Oc3ncccn3)[C@@H](F)C2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
IRAK4 Q9NWZ3 4/20 0.39
PIM1 P11309 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 1/20 0.36
PTK2 Q05397 1/20 0.36
HPGD P15428 1/20 0.36
GRM4 Q14833 1/20 0.36
GPR6 P46095 1/20 0.35
KDM4E B2RXH2 1/20 0.35
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
OPRK1 P41145 1/20 0.34
P2RX7 Q99572 1/20 0.34
TYK2 P29597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13634544 1.00 MEN1 (0.40) MEN1KMT2AIRAK4PIM1SMN1; SMN2
SCHEMBL13634631 0.95 GPR6 (0.40) MEN1KMT2AIRAK4PIM1GRM4
SCHEMBL13634630 0.95 GPR6 (0.40) MEN1KMT2AIRAK4PIM1GRM4
SCHEMBL13634622 0.92 PIM1 (0.48) MEN1KMT2AIRAK4PIM1GPR6
SCHEMBL13634787 0.88 HCAR2 (0.40) MEN1KMT2AIRAK4SMN1; SMN2ALDH1A1
SCHEMBL13270803 0.88 HCAR2 (0.40) MEN1KMT2AIRAK4SMN1; SMN2ALDH1A1
SCHEMBL13634623 0.88 PIM1 (0.44) IRAK4PIM1GRM4GPR6
SCHEMBL13634890 0.87 ALDH1A1 (0.37) KMT2AIRAK4SMN1; SMN2ALDH1A1HPGD
SCHEMBL13634860 0.87 POLB (0.43) KMT2ASMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL13634726 0.86 GPR6 (0.38) MEN1KMT2AIRAK4ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed