SCHEMBL13634882

SCHEMBL13634882

O=C(Nc1ccc(C(=O)N2CCS(=O)(=O)CC2)cc1Br)c1csc(N2CCC(Oc3ncccn3)CC2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K7 O43318 1/20 0.39
SCD O00767 1/20 0.36
PRSS12 P56730 2/20 0.36
GPR6 P46095 2/20 0.36
CHEK1 O14757 2/20 0.35
PIM1 P11309 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC2 Q92769 1/20 0.34
NPC1 O15118 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
GRM4 Q14833 1/20 0.34
LRRK2 Q5S007 2/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13634863 0.92 MAP3K7 (0.48) MAP3K7SCDGPR6
SCHEMBL13634880 0.89 RAB9A (0.40) MAP3K7SCDPRSS12PIM1NPC1
SCHEMBL13634653 0.88 HRH3 (0.41) SCDGPR6CHEK1HDAC3HDAC2
SCHEMBL13634849 0.88 GPR6 (0.41) SCDGPR6CHEK1PIM1HDAC3
SCHEMBL13634547 0.87 MAP3K7 (0.39) MAP3K7SCDPRSS12GPR6PIM1
SCHEMBL13634881 0.87 NPC1 (0.40) SCDGPR6CHEK1PIM1HDAC3
SCHEMBL13634828 0.85 RAB9A (0.41) SCDPIM1NPC1MAPTRAB9A
SCHEMBL13634698 0.83 MAP3K7 (0.47) MAP3K7SCDGPR6
SCHEMBL13634648 0.83 MAP3K7 (0.51) MAP3K7GPR6CHEK1LRRK2
SCHEMBL13634883 0.82 NPC1 (0.43) CHEK1PIM1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed