SCHEMBL13650809

SCHEMBL13650809

C1=CCCC(N2CCNCC2)=C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
ADRB1 P08588 7/20 0.36
HTR3E A5X5Y0 2/20 0.36
HTR3B O95264 2/20 0.36
HTR3A P46098 2/20 0.36
HTR3D Q70Z44 2/20 0.36
HTR3C Q8WXA8 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
HRH1 P35367 1/20 0.36
USP2 O75604 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CASP1 P29466 1/20 0.35
CASP4 P49662 1/20 0.35
CASP5 P51878 1/20 0.35
ADRB2 P07550 2/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM1 P11229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17934702 0.79
SCHEMBL18052759 0.79 ADRB1 (0.41) ALDH1A1KDM4EADRB1HTR3EHTR3B
SCHEMBL29980540 0.76 ADRA2C (0.34) ALDH1A1KDM4EHTR3EHTR3BHTR3A
SCHEMBL30425332 0.76 LMNA (0.36) ALDH1A1KDM4EUSP2LMNA
SCHEMBL20483904 0.72 ADRB1 (0.47) ALDH1A1KDM4EADRB1HTR3EHTR3B
SCHEMBL19120784 0.72 MAPT (0.46) ALDH1A1ADRB1HTR3EHTR3BHTR3A
SCHEMBL20780839 0.72
SCHEMBL12663101 0.72 CHRNA7 (0.42) ALDH1A1KDM4EUSP2SMN1; SMN2LMNA
SCHEMBL31696522 0.71 ALDH1A1 (0.33) ALDH1A1
SCHEMBL1709261 0.71 NPC1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113214287-B HPK1 inhibitors and methods of use thereof 大学健康网络 2023-10-20 CN disclosed
US-20170290825-A1 PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY AGIOS PHARMACEUTICALS, INC. 2017-10-12 US disclosed
WO-2009123221-A1 PYRIMIDINE DERIVATIVE HAVING CELL-PROTECTING ACTIVITY AND USE THEREOF 全薬工業株式会社 (JP) 2009-10-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170290825-A1 PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY PCK1, PDK3, PDK2 ALDH1A1 1517/4885KDM4E 2079/4885ADRB1 3032/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.