SCHEMBL13668590

SCHEMBL13668590

N#Cc1ccc2nc(O)cnc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.40
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
CA3 P07451 1/20 0.38
CA6 P23280 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
HPGDS O60760 1/20 0.37
MAP4K4 O95819 3/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
DYRK1A Q13627 1/20 0.36
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36
HSD17B14 Q9BPX1 1/20 0.36
PKN1 Q16512 1/20 0.36
PKN2 Q16513 1/20 0.36
APP P05067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13668594 0.93 PIN1 (0.40) PIN1CA12CA2CA3CA6
SCHEMBL1035242 0.79 ALDH1A1 (0.47) PIN1CA2HPGDSKDM4EALDH1A1
SCHEMBL6422468 0.79 GRM5 (0.42) HPGDSKDM4EALDH1A1CYP11B1CYP11B2
SCHEMBL4726210 0.79 CDC7 (0.41) PIN1HPGDSMAP4K4KDM4EALDH1A1
SCHEMBL2437956 0.77 PIN1 (0.44) PIN1CA12CA2CA3CA6
SCHEMBL14582923 0.75 ESR2 (0.48) MAP4K4KDM4EALDH1A1GAADYRK1A
SCHEMBL25260514 0.74 HRH3 (0.46) PIN1CA12CA2CA3CA6
SCHEMBL622637 0.72 CDK5 (0.47) PIN1MAP4K4KDM4EALDH1A1GLA
SCHEMBL15197891 0.72 PIN1 (0.42) PIN1CA2KDM4EALDH1A1GLA
SCHEMBL30189727 0.72 HPGD (0.45) MAP4K4KDM4EALDH1A1GAAMETAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180155341-A1 Antibacterial Compounds JANSSEN SCIENCES IRELAND UC (IE) 2018-06-07 US disclosed
WO-2017001661-A1 ANTIBACTERIAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2017-01-05 WO disclosed
US-20090258862-A1 Niacin receptor agonists, compositions containing such compounds and methods of treatment MERCK SHARP & DOHME CORP. 2009-10-15 US disclosed
WO-2007027532-A2 NIACIN RECEPTOR AGONISTS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK & CO., INC. (US) 2007-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090258862-A1 Niacin receptor agonists, compositions containing such compounds and methods of treatment LDLR, APOB, FFAR1 PIN1 4694/4885CA12 4768/4885CA2 4250/4885
US-20180155341-A1 Antibacterial Compounds FDPS, SQOR, NDUFS3 PIN1 524/4885CA12 4157/4885CA2 3368/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.