SCHEMBL13680483

SCHEMBL13680483

Cc1cccc(-c2ccc(NC(=O)N(C)C)cc2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
PNPLA2 Q96AD5 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
MAPT P10636 2/20 0.45
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
NFKB1 P19838 1/20 0.45
STAT1 P42224 1/20 0.45
RAB9A P51151 1/20 0.45
NFKB2 Q00653 1/20 0.45
KMT2A Q03164 1/20 0.45
RELA Q04206 1/20 0.45
GBA1 P04062 1/20 0.44
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
AOC3 Q16853 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12270039 0.83 KMT2A (0.61) MAPTMEN1NPC1NFKB1STAT1
SCHEMBL13680585 0.82 KIF11 (0.56) MAPTMEN1NPC1NFKB1STAT1
SCHEMBL13537053 0.81 SMN1; SMN2 (0.49) TSHRMAPTMEN1NPC1NFKB1
SCHEMBL13680553 0.81 GBA1 (0.52) TSHRMAPTMEN1NPC1NFKB1
SCHEMBL11686928 0.77 SMN1; SMN2 (0.48) TSHRMAPTMEN1NPC1RAB9A
SCHEMBL13680473 0.77 TGFBR1 (0.48) TSHRMEN1KMT2ATP53SMN1; SMN2
SCHEMBL13680841 0.77 TSHR (0.40) TSHRPNPLA2HDAC6MEN1KMT2A
SCHEMBL13680672 0.76 CYP1A2 (0.46) TSHRMAPTMEN1NPC1NFKB1
SCHEMBL3422361 0.75 CCR1 (0.75) MAPTMEN1RAB9AKMT2A
SCHEMBL687878 0.75 TSHR (0.79) TSHRMEN1KMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed