SCHEMBL13680722

SCHEMBL13680722

Cc1ccc(-c2cnc(N3CCNCC3)nc2)o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.44
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPKAPK2 P49137 4/20 0.39
MAPT P10636 1/20 0.39
HTR2C P28335 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
CYP1A2 P05177 4/20 0.39
CYP2C19 P33261 3/20 0.39
HPGD P15428 3/20 0.39
CASP1 P29466 3/20 0.39
CASP7 P55210 3/20 0.39
HSD17B10 Q99714 3/20 0.39
CYP3A4 P08684 2/20 0.39
TSHR P16473 1/20 0.39
ADRB1 P08588 1/20 0.38
GHSR Q92847 1/20 0.38
USP2 O75604 1/20 0.37
GLA P06280 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680712 0.86 NPY5R (0.40) ALDH1A1KDM4EMAPTCYP1A2CYP2C19
SCHEMBL13680708 0.84 CNR2 (0.48) KDM4E
SCHEMBL4582837 0.75 HTR1A (0.54) TAAR1ALDH1A1KDM4EMAPTCHRNB2
SCHEMBL7991455 0.73 ALDH1A1 (0.59) TAAR1ALDH1A1KDM4ECHRNB2CHRNA4
Hydrochloric Acid SCHEMBL28966659 0.72 ALDH1A1 (0.62) TAAR1ALDH1A1KDM4ECHRNB2CHRNA4
SCHEMBL13680715 0.71 TDP1 (0.42) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL9400977 0.71 TAAR1 (0.64) TAAR1ALDH1A1KDM4ECYP1A2CYP2C19
SCHEMBL4582036 0.71 ADRB1 (0.54) TAAR1ALDH1A1KDM4EHTR2CCYP1A2
SCHEMBL13680685 0.70 KCNH2 (0.49) TAAR1ALDH1A1KDM4EMAPTCYP1A2
SCHEMBL6787637 0.69 HTR7 (0.54) TAAR1ALDH1A1KDM4ECYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed