SCHEMBL13680855

SCHEMBL13680855

Cn1ncc2cc(-c3cccc(CCC=O)n3)ccc21

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 7/20 0.42
TRPA1 O75762 1/20 0.42
TGFBR1 P36897 7/20 0.39
MAPK14 Q16539 6/20 0.39
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39
CREBBP Q92793 2/20 0.38
BRD4 O60885 1/20 0.37
AR P10275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680984 0.78 LMNA (0.39) IRAK4TRPA1CCNCCDK8CREBBP
SCHEMBL13680555 0.75 TGFBR1 (0.55) IRAK4TRPA1TGFBR1MAPK14
SCHEMBL13680907 0.75 APP (0.42) TRPA1CCNCCDK8CREBBPBRD4
SCHEMBL15332767 0.74 TRPA1 (0.49) TRPA1TGFBR1MAPK14CREBBPBRD4
SCHEMBL17547051 0.74 TRPA1 (0.49) TRPA1TGFBR1MAPK14CCNCCDK8
SCHEMBL13680834 0.74 PDE10A (0.39) IRAK4
SCHEMBL13680847 0.73 PDE10A (0.43) IRAK4
SCHEMBL13680817 0.73 ALDH1A1 (0.47)
SCHEMBL15341838 0.72 TRPA1 (0.47) IRAK4TRPA1
SCHEMBL3854280 0.72 MEN1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed