SCHEMBL13680901

SCHEMBL13680901

O=CCCc1ccc(-c2ccc(OC(F)(F)F)nc2)o1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.36
CYP2C19 P33261 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
PRMT1 Q99873 2/20 0.33
ALDH1A1 P00352 6/20 0.32
MAPT P10636 4/20 0.32
PKM P14618 4/20 0.32
KDM4E B2RXH2 3/20 0.32
PPARD Q03181 2/20 0.32
CYP2A6 P11509 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680900 0.84 MAPT (0.41) ALDH1A1MAPTPKMKDM4ECYP2A6
SCHEMBL13680885 0.81 TRPV4 (0.35) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL13680868 0.81 PRMT1 (0.49) CYP1A2CYP2C19CYP2C9PRMT1ALDH1A1
SCHEMBL13680889 0.79 ALDH1A1 (0.36) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL13680899 0.77 CYP2C19 (0.40) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL13680956 0.74 SHMT2 (0.40) ALDH1A1MAPTKDM4EPPARDHPGD
SCHEMBL13681294 0.73 ALDH1A1 (0.33) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL13680902 0.73 APP (0.40) CYP1A2CYP2C19ALDH1A1MAPTPKM
SCHEMBL13680896 0.73 ALDH1A1 (0.41) CYP1A2CYP2C19CYP3A4PRMT1ALDH1A1
SCHEMBL13681006 0.73 CYP2C19 (0.39) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed