SCHEMBL1368532

SCHEMBL1368532

CN(C)C(=O)c1cccc(Br)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.57
ALDH1A1 P00352 3/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
TP53 P04637 1/20 0.50
LMNA P02545 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
POLB P06746 1/20 0.49
MAPT P10636 1/20 0.49
ALPG P10696 1/20 0.49
ATM Q13315 1/20 0.49
TLR9 Q9NR96 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
HPGD P15428 1/20 0.47
C1S P09871 1/20 0.47
CDK4 P11802 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29852161 1.00 PARP1 (0.57) PARP1ALDH1A1L3MBTL1TP53LMNA
SCHEMBL17758892 0.86 PARP1 (0.55) PARP1ALDH1A1L3MBTL1TP53LMNA
SCHEMBL7406706 0.85 MEN1 (0.55) ALDH1A1L3MBTL1MEN1KMT2AATM
SCHEMBL3931604 0.82 PARP1 (0.44) PARP1ALDH1A1L3MBTL1LMNAMEN1
SCHEMBL935497 0.82 PARP1 (0.50) PARP1ALDH1A1L3MBTL1TP53LMNA
SCHEMBL8366933 0.82 CDK4 (0.52) PARP1ALDH1A1L3MBTL1TP53LMNA
SCHEMBL4300450 0.81 HPGD (0.69) PARP1ALDH1A1L3MBTL1LMNAMAPT
SCHEMBL6177291 0.80 KDM1A (0.56) PARP1ALDH1A1L3MBTL1LMNAMEN1
SCHEMBL14095771 0.80 ALDH1A1 (0.41) PARP1ALDH1A1TP53NPSR1CYP1A2
SCHEMBL7455084 0.79 HSD17B2 (0.47) PARP1ALDH1A1L3MBTL1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 115 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260132132-A1 3A,4,5,6-TETRAHYDRO-1 H-PYRAZOLO[3,4-C]PYRIDIN-7(7AH)-ONE DERIVATIVES AS FACTOR XIIA INHIBITORS KALVISTA PHARMACEUTICALS LTD (GB) 2026-05-14 US disclosed
EP-4051667-B1 HETEROCYCLIC CARBOXYLATE COMPOUNDS AS GLYCOLATE OXIDASE INHIBITORS LILAC THERAPEUTICS INC (US) 2026-01-28 EP disclosed
US-12398139-B2 Modulators of AMPA receptor signaling CENTRE FOR ADDICTION AND MENTAL HEALTH (CA) 2025-08-26 US disclosed
CN-117342963-B 1, 4-Dicarbonyl compound, and preparation method and application thereof 上海予君生物科技发展有限公司 2025-06-17 CN disclosed
EP-3935059-B1 MODULATORS OF AMPA RECEPTOR SIGNALING CAMH (CA) 2025-04-23 EP disclosed
US-20250064787-A1 Heterocyclic Carboxylate Compounds as Glycolate Oxidase Inhibitors LILAC THERAPEUTICS INC (US) 2025-02-27 US disclosed
US-12168002-B2 Heterocyclic carboxylate compounds as glycolate oxidase inhibitors Lilac Therapeutics, Inc. (US) 2024-12-17 US disclosed
EP-4470538-A2 HETEROCYCLIC CARBOXYLATE COMPOUNDS AS GLYCOLATE OXIDASE INHIBITORS Lilac Therapeutics, Inc. (US) 2024-12-04 EP disclosed
WO-2024175081-A1 SHP2 INHIBITOR COMPOUND AND USE THEREOF 深圳真实生物医药科技有限公司 2024-08-29 WO disclosed
US-11970499-B1 Pyrazolo[1,5-c]pyrimidine compounds as CK2 inhibitors King Faisal University (SA) 2024-04-30 US disclosed
EP-0284076-B1 Process for preparing (+)-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds SYNTEX INC (US) 1994-06-08 EP disclosed
WO-1993021178-A1 INDOLE DERIVATIVES AS 5-HT1-LIKE AGONISTS PFIZER LIMITED (GB) 1993-10-28 WO disclosed
EP-0275092-B1 PROCESS FOR PREPARING (+)-1,2-DIHYDRO-3H-PYRROLO(1,2-A)PYRROLE-1,7-DICARBOXYLATES SYNTEX (U.S.A.) INC. (US) 1992-06-03 EP disclosed
EP-0284076-A1 Process for preparing (+)-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds SYNTEX (U.S.A.) INC. (US) 1988-09-28 EP disclosed
EP-0275092-A1 Process for preparing (+)-1,2-dihydro-3H-pyrrolo(1,2-a)pyrrole-1,7-dicarboxylates SYNTEX (U.S.A.) INC. (US) 1988-07-20 EP disclosed
EP-0041711-B1 6-CHLORO- OR 6-BROMO-1,2-DIHYDRO-3H-PYRROLO(1,2-A)-PYRROLE-1-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF, PROCESS FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SYNTEX (U.S.A.) INC. (US) 1985-04-17 EP disclosed
US-4410534-A 3-Substituted-5,6,7,8-tetrahydropyrrolo[1,2-a]-pyridine-and 6,7,8,9-tetrahydro-5H-pyrrolo[1,2-a]-azepine carboxylic acid derivatives useful as blood platelet aggregation inhibitors SYNTEX (U.S.A.) INC. (US) 1983-10-18 US disclosed
US-4344943-A ANALGESICS, ANTIINFLAMMATORY AGENTS SYNTEX (U.S.A.) INC. (US) 1982-08-17 US disclosed
EP-0041711-A1 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo(1,2-a)-pyrrole-1-carboxylic acids and derivatives thereof, process for their production and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1981-12-16 EP disclosed
US-4089969-A ANTIINFLAMMATORY, ANALGESIC, ANTIPYRETIC, SMOOTH MUSCLE RELAXANT SYNTEX (U.S.A.) INC. (US) 1978-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260132132-A1 3A,4,5,6-TETRAHYDRO-1 H-PYRAZOLO[3,4-C]PYRIDIN-7(7AH)-ONE DERIVATIVES AS FACTOR XIIA INHIBITORS F11, F13B, F7 PARP1 462/4885ALDH1A1 2202/4885L3MBTL1 3267/4885
US-12168002-B2 Heterocyclic carboxylate compounds as glycolate oxidase inhibitors UGDH, PGD, PNPO PARP1 2506/4885ALDH1A1 184/4885L3MBTL1 3238/4885
US-11970499-B1 Pyrazolo[1,5-c]pyrimidine compounds as CK2 inhibitors CDK2, TK1, CDK1 PARP1 1349/4885ALDH1A1 4311/4885L3MBTL1 3656/4885
US-12398139-B2 Modulators of AMPA receptor signaling GRM2, GRM1, GRIK1 PARP1 3947/4885ALDH1A1 1697/4885L3MBTL1 3511/4885
US-20250064787-A1 Heterocyclic Carboxylate Compounds as Glycolate Oxidase Inhibitors GLS, DUOX1, HAO1 PARP1 1582/4885ALDH1A1 100/4885L3MBTL1 1957/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.