SCHEMBL13988024

SCHEMBL13988024

Cc1ccccc1CCN(CCCCC(=O)c1ccc2c(c1)CCC(=O)N2)C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.43
HTR2A P28223 2/20 0.43
HTR7 P34969 2/20 0.43
DRD3 P35462 2/20 0.43
DRD4 P21917 1/20 0.43
DRD2 P14416 2/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
HDAC3 O15379 2/20 0.38
HDAC4 P56524 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HDAC9 Q9UKV0 2/20 0.38
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
GRIN2B Q13224 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4856265 0.91 HTR1A (0.42) HTR1AHTR2AHTR7DRD3DRD4
SCHEMBL4852226 0.90 ACHE (0.42) HTR1AHTR2AHTR7DRD3DRD4
SCHEMBL4861872 0.90 MAOA (0.47) HTR1AHTR2AHTR7DRD3DRD4
SCHEMBL13987983 0.84 NPSR1 (0.47)
SCHEMBL13988041 0.83 CYP11B1 (0.36) DRD2GRIN2B
SCHEMBL13988010 0.83 ALDH1A1 (0.48)
SCHEMBL13988032 0.81 HDAC1 (0.33) HDAC3HDAC1HDAC2
SCHEMBL13988043 0.80 CTNNB1 (0.35) HDAC3HDAC1HDAC2
SCHEMBL4851846 0.80 DRD3 (0.44) HTR1AHTR2AHTR7DRD3DRD4
SCHEMBL4858283 0.78 HTR1A (0.46) HTR1AHTR2AHTR7DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7462628-B2 Preventives/remedies for urinary disturbance TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-12-09 US disclosed