SCHEMBL14064862

SCHEMBL14064862

CC(C)(C)C(CC#N)OC(=O)NCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.48
CTSS P25774 4/20 0.44
CTSL P07711 3/20 0.44
CTSB P07858 3/20 0.44
CTSK P43235 3/20 0.44
RIPK1 Q13546 1/20 0.43
CASP3 P42574 1/20 0.42
UTS2R Q9UKP6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28614724 0.82 MCL1 (0.51) MCL1CASP3UTS2R
SCHEMBL28603794 0.82 MCL1 (0.51) MCL1CASP3UTS2R
SCHEMBL28919836 0.81 IMPDH2 (0.56) CTSLCTSBCTSK
SCHEMBL451232 0.81 MTNR1A (0.42) CTSSCTSBCTSK
SCHEMBL28601403 0.80 MCL1 (0.49) MCL1CTSSCTSLCTSBCTSK
SCHEMBL27549418 0.78 OPRM1 (0.46) RIPK1
SCHEMBL19509288 0.77 RAB9A (0.51) RIPK1CASP3
SCHEMBL28600675 0.77 MCL1 (0.48) MCL1CASP3
SCHEMBL28600679 0.76 MCL1 (0.50) MCL1CASP3
SCHEMBL20354607 0.74 KMT2A (0.53) CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1964561-A1 Inhibitors of IMPDH enzyme Vertex Pharmaceuticals Incorporated (US) 2008-09-03 EP disclosed