SCHEMBL14200380

SCHEMBL14200380

CCCC1Cc2ccccc2N1C(=O)CC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.47
PKM P14618 1/20 0.46
DRD2 P14416 7/20 0.45
DRD4 P21917 7/20 0.45
ALDH1A1 P00352 5/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 2/20 0.44
NPC1 O15118 1/20 0.44
CYP2D6 P10635 1/20 0.44
MEN1 O00255 1/20 0.41
CYP3A4 P08684 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200379 0.87 MTNR1A (0.50) PKMMEN1KMT2A
SCHEMBL24201848 0.86 DRD2 (0.53) NOTUMPKMDRD2DRD4ALDH1A1
SCHEMBL14229140 0.85 NOTUM (0.50) NOTUMPKMDRD2DRD4ALDH1A1
SCHEMBL7593171 0.74 NOTUM (0.57) NOTUMPKMDRD2DRD4ALDH1A1
SCHEMBL7067724 0.74 MTNR1A (0.43) PKMALDH1A1MEN1KMT2A
SCHEMBL5556232 0.73 PKM (0.51) NOTUMPKMALDH1A1CYP1A2CYP2C19
SCHEMBL18701883 0.72 DRD2 (0.51) NOTUMPKMDRD2DRD4ALDH1A1
SCHEMBL14229139 0.72 MTNR1A (0.48) PKM
SCHEMBL14200385 0.71 MTNR1A (0.43) NOTUMALDH1A1CYP1A2CYP2C19NPC1
SCHEMBL27968682 0.70 NOTUM (0.52) NOTUMPKMDRD2DRD4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed