SCHEMBL1426486

SCHEMBL1426486

COc1ccc2c(c1O)C(=O)c1ccccc1C2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 1.00
MEN1 O00255 6/20 1.00
KMT2A Q03164 6/20 1.00
RAB9A P51151 4/20 1.00
NPC1 O15118 3/20 1.00
SMN1; SMN2 Q16637 4/20 0.68
ALDH1A1 P00352 4/20 0.65
KDM4E B2RXH2 3/20 0.65
USP2 O75604 1/20 0.65
DUSP3 P51452 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
ELANE P08246 5/20 0.62
MAPK1 P28482 2/20 0.61
CYP3A4 P08684 1/20 0.61
BCL2 P10415 1/20 0.61
HPGD P15428 1/20 0.61
ALOX15 P16050 1/20 0.61
ALOX12 P18054 1/20 0.61
MAOA P21397 1/20 0.61
APEX1 P27695 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29929605 1.00 MAPT (1.00) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL31441205 1.00 MAPT (1.00) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL3276344 0.85 MAPT (0.74) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL3959473 0.82 MAPT (0.69) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL23199010 0.81 MAPT (0.69) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL28206847 0.81 MEN1 (0.69) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL496978 0.81 RAB9A (1.00) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL30030177 0.80 ADORA2A (0.68) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL3955390 0.80 MAPT (0.67) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL27715756 0.80 MAPT (0.67) MAPTMEN1KMT2ARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240315965-A1 COMPOSITIONS AND METHODS RELATED TO PHARMACEUTICAL EXCIPIENTS Natural Extraction Systems, LLC (US) 2024-09-26 US claimed
US-20230089351-A1 METHODS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES Natural Extraction Systems, LLC (US) 2023-03-23 US claimed
WO-2022182523-A1 COMPOSITIONS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES Natural Extraction Systems, LLC (US) 2022-09-01 WO claimed
WO-2022182527-A1 COMPOSITIONS AND METHODS RELATED TO PHARMACEUTICAL EXCIPIENTS Natural Extraction Systems, LLC (US) 2022-09-01 WO claimed
EP-3943085-A2 TOMM6-INTERACTING EXTRACTS AND COMPOUNDS FOR USE IN THE TREATMENT AND PROPHYLAXIS OF NERVOUS SYSTEM DISEASES, ATHEROSCLEROSIS, HEPATITIS B INFECTION AND HUMAN PAPILLOMA VIRUS (HPV) INFECTION ETH Zurich (CH) 2022-01-26 EP claimed
WO-2021158575-A1 COMPOSITIONS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES Natural Extraction Systems, LLC (US) 2021-08-12 WO claimed
WO-2021158573-A1 METHODS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES Natural Extraction Systems, LLC (US) 2021-08-12 WO claimed
US-20210186947-A1 TOMM6-INTERACTING EXTRACTS AND COMPOUNDS FOR USE IN THE TREATMENT AND PROPHYLAXIS OF NERVOUS SYSTEM DISEASES, ATHEROSCLEROSIS, HEPATITIS B INFECTION AND HUMAN PAPILLOMA VIRUS (HPV) INFECTION ETH ZURICH (CH) 2021-06-24 US claimed
EP-3801507-A2 TOMM6-INTERACTING EXTRACTS AND COMPOUNDS FOR USE IN THE TREATMENT AND PROPHYLAXIS OF NERVOUS SYSTEM DISEASES, ATHEROSCLEROSIS, HEPATITIS B INFECTION AND HUMAN PAPILLOMA VIRUS (HPV) INFECTION ETH Zurich (CH) 2021-04-14 EP claimed
WO-2010079914-A2 A COMPOSITION COMPRISING THE COMPOUND ISOLATED FROM THE EXTRACT OF RUBIAE RADIX FOR PREVENTING AND TREATING INFLAMMATORY DISEASES INDUSTRY-ACADEMIC COORPERATION FOUNDATION DAEGU HAANY UNIVERSITY (KR) 2010-07-15 WO claimed
US-20260048025-A1 COMPOSITIONS AND METHODS RELATED TO DISSOLVED OXIDES NATURAL EXTRACTION SYS LLC (US) 2026-02-19 US disclosed
US-12409152-B2 Compositions and methods related to dissolved oxides Natural Extraction Systems, LLC (US) 2025-09-09 US disclosed
US-20250161394-A1 Compositions Comprising Kavalactones NATURAL EXTRACTION SYS LLC (US) 2025-05-22 US disclosed
US-20240315965-A1 COMPOSITIONS AND METHODS RELATED TO PHARMACEUTICAL EXCIPIENTS Natural Extraction Systems, LLC (US) 2024-09-26 US disclosed
CN-108700808-B Masking resist composition for etching, method for producing substrate using same, and method for producing light-emitting element 东丽株式会社 2024-04-05 CN disclosed
WO-2009060017-A1 HAIR TREATMENT AGENT COMPRISING TILIROSIDE AND VITAMIN B HENKEL AG & CO. KGAA (DE) 2009-05-14 WO disclosed
WO-2009033833-A2 COLORING AGENT HAVING NATURAL DYES AND 1,3-DIHYDROXYACETONE HENKEL AG & CO. KGAA (DE) 2009-03-19 WO disclosed
WO-2008100977-A2 CARBAMATES THERAPEUTIC RELEASE AGENTS AS AMIDASE INHIBITORS N.V. ORGANON (NL) 2008-08-21 WO disclosed
US-4346103-A MULTIPLE SCLEROSIS FRIEDMANN CHARLES A 1982-08-24 US disclosed
US-4244968-A HYDROXY- AND AMINO-ANTHRAQUINONES PROTER S.P.A. (IT) 1981-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230089351-A1 METHODS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES FABP2, FABP4, GUSB MAPT 3926/4885MEN1 1711/4885KMT2A 4742/4885
US-12409152-B2 Compositions and methods related to dissolved oxides PRKG2, PRKG1, CIT MAPT 2118/4885MEN1 593/4885KMT2A 3932/4885
US-20210186947-A1 TOMM6-INTERACTING EXTRACTS AND COMPOUNDS FOR USE IN THE TREATMENT AND PROPHYLAXIS OF NERVOUS SYSTEM DISEASES, ATHEROSCLEROSIS, HEPATITIS B INFECTION AND HUMAN PAPILLOMA VIRUS (HPV) INFECTION TOMM70, TOMM34, TIMM50 MAPT 2071/4885MEN1 2055/4885KMT2A 4561/4885
US-20260048025-A1 COMPOSITIONS AND METHODS RELATED TO DISSOLVED OXIDES SCO2, CNR2, CNR1 MAPT 3552/4885MEN1 1906/4885KMT2A 4414/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.