SCHEMBL6974600

SCHEMBL6974600

CC(C)c1nc(COCc2ccccc2)[nH]c1Sc1cc(F)cc(F)c1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
DHODH Q02127 1/20 0.33
MAPK14 Q16539 1/20 0.32
VCP P55072 1/20 0.32
CAPN1 P07384 1/20 0.32
TACR1 P25103 1/20 0.31
PDE9A O76083 1/20 0.31
PDE1A P54750 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE1C Q14123 1/20 0.31
ALDH1A1 P00352 2/20 0.30
ALOX5 P09917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14439826 0.88 TSHR (0.39) TSHRVCPCAPN1PDE9APDE1A
SCHEMBL5852619 0.87 TACR1 (0.34) TSHRDHODHVCPCAPN1TACR1
SCHEMBL6964698 0.83 LMNA (0.36) TACR1PDE9APDE1APDE1BPDE1C
SCHEMBL5029294 0.83 DHFR (0.41) ALDH1A1
SCHEMBL14439851 0.81 TSHR (0.41) TSHRDHODHVCPCAPN1PDE9A
SCHEMBL6971891 0.78 ALDH1A1 (0.37) DHODHCAPN1TACR1ALDH1A1
SCHEMBL6962115 0.76 ADRB2 (0.32) MAPK14CAPN1
SCHEMBL6962307 0.76 CYP1A2 (0.35) DHODHALDH1A1
SCHEMBL6971468 0.76 HRH4 (0.36) CAPN1TACR1ALDH1A1
SCHEMBL8494052 0.75 CYP19A1 (0.37) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed