SCHEMBL14560403

SCHEMBL14560403

CC(=O)OCCc1c(C=O)[nH]c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.48
HTR6 P50406 2/20 0.42
MAPT P10636 2/20 0.41
TSHR P16473 2/20 0.41
HKDC1 Q2TB90 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
HTR1F P30939 1/20 0.41
HTR7 P34969 1/20 0.41
DRD3 P35462 1/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27817269 0.82 ALDH1A1 (0.60) RAD52HTR6MAPTTSHRHTR1A
SCHEMBL14560412 0.78 MTNR1A (0.65) MAPTTSHRMEN1CYP1A2CYP3A4
SCHEMBL28804680 0.78 RAB9A (0.54) HTR6MAPTTSHRHKDC1NPSR1
SCHEMBL14560402 0.77 KDM4E (0.64) MAPTHKDC1NPSR1MEN1KMT2A
SCHEMBL14560404 0.77 EGFR (0.62) HTR6MAPTHKDC1NPSR1ALDH1A1
SCHEMBL13962342 0.76 SIRT1 (0.48) RAD52HTR6MAPTTSHRMEN1
SCHEMBL14560406 0.76 EGFR (0.66) HTR6MAPTHKDC1NPSR1HTR1A
SCHEMBL14560419 0.76 KDM4E (0.62) HTR6MAPTTSHRHKDC1NPSR1
SCHEMBL28204517 0.75 MAPT (0.41) HTR6MAPTTSHRHKDC1NPSR1
SCHEMBL7380422 0.75 HTT (0.51) MAPTTSHRHKDC1NPSR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189721-B2 Bicyclic protein kinase inhibitors SUGEN INC. (US) 2007-03-13 US disclosed
US-7189721-B2 Bicyclic protein kinase inhibitors SUGEN INC. (US) 2007-03-13 US disclosed